SCHEMBL289044

SCHEMBL289044

N[C@@H](Cc1c[nH]c2ccccc12)C(=O)OC(=O)[C@@H](N)Cc1c[nH]c2ccccc12

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.74
KDM4E B2RXH2 2/20 0.74
MEN1 O00255 2/20 0.74
LMNA P02545 2/20 0.74
KMT2A Q03164 2/20 0.74
MPO P05164 1/20 0.74
TSHR P16473 1/20 0.74
BLM P54132 1/20 0.74
PMP22 Q01453 1/20 0.74
HIF1A Q16665 1/20 0.74
TACR1 P25103 2/20 0.66
HTR2A P28223 2/20 0.59
ADRB1 P08588 1/20 0.59
HTR1A P08908 1/20 0.59
ADRA2A P08913 1/20 0.59
SLC6A2 P23975 1/20 0.59
HTR1D P28221 1/20 0.59
HTR1B P28222 1/20 0.59
HTR2C P28335 1/20 0.59
HTR1E P28566 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL475351 1.00 MAPT (0.74) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL27645874 0.95 MAPT (0.67) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL4261073 0.95 MAPT (0.67) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL21059260 0.94 MAPT (0.70) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL120931 0.93 KDM4E (0.69) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL8406415 0.93 MAPT (0.65) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL5065255 0.93 KDM4E (0.65) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL17503190 0.93 MAPT (0.72) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL1640627 0.93 MAPT (0.68) MAPTKDM4EMEN1LMNAKMT2A
SCHEMBL626831 0.93 MAPT (0.72) MAPTKDM4EMEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1637185-B1 Controlled-release formulations containing tryptophan and/or 5-hydroxytryptophan AMBROS PHARMA S R L (IT) 2008-08-20 EP claimed
US-5892112-A ACYLATION OF AMINO ACIDS WITH ANHYDRIDES OR CARBOXY GROUPS, AMIDATION WITH AMINE AND CONVERSION OF ACID OR ESTER TO HYDROXAMIC ACID AND HYDROLYSIS GLYCOMED INCORPORATED (US) 1999-04-06 US claimed
CN-115304661-B Cyclic peptide compound and application thereof 西南民族大学 2024-03-15 CN disclosed
CN-107304191-B Indolylamine 2,3-dioxygenase inhibitor and preparation method and application thereof 上海翰森生物医药科技有限公司 2023-09-29 CN disclosed
CN-111491923-B N- (2-cyclohexylethyl) carboxamide derivatives, preparation and pharmaceutical use thereof 上海海雁医药科技有限公司 2023-06-16 CN disclosed
WO-2023088591-A1 BACTERIAL STRAIN AND THE USE THEREOF PROBITAT OY (FI) 2023-05-25 WO disclosed
CN-112384502-B Cycloalkyl-substituted amide derivatives, preparation method and medical application thereof 上海海雁医药科技有限公司 2022-11-08 CN disclosed
CN-106883193-B Indoleamine 2,3-dioxygenase inhibitor as well as preparation method and application thereof 上海翰森生物医药科技有限公司 2021-10-15 CN disclosed
CN-108424944-B Optimized production method and culture medium of candicidin 华东理工大学 2021-07-27 CN disclosed
CN-112384502-A Cycloalkyl-substituted amide derivatives, preparation method and medical application thereof 上海海雁医药科技有限公司 2021-02-19 CN disclosed
CN-110105275-B Amide derivatives, preparation method and medical application thereof 上海海雁医药科技有限公司 2020-12-29 CN disclosed
CN-101969984-A Haemostasis- modulating compositions and uses therefor UNIV QUEENSLAND 2011-02-09 CN disclosed
WO-2011000753-A1 METHOD FOR NORMALIZATION IN METABOLOMICS ANALYSIS METHODS WITH ENDOGENOUS REFERENCE METABOLITES BIOCRATES LIFE SCIENCES AG (AT) 2011-01-06 WO disclosed
WO-2010128054-A1 METHOD OF DIAGNOSING ASPHYXIA BIOCRATES LIFE SCIENCES AG (AT) 2010-11-11 WO disclosed
WO-2010075287-A2 COMPOUNDS AND METHODS FOR THE TREATMENT OF PAIN AND OTHER DISEASES AQUILUS PHARMACEUTICALS, INC (US) 2010-07-01 WO disclosed
CN-101541379-A Methods for modulating cell survival INST MEDICAL W & E HALL (AU) 2009-09-23 CN disclosed
CN-1938042-A Methods for mitigating oxidative damage CORNELL RES FOUNDATION INC (US) 2007-03-28 CN disclosed
US-5460725-A Crosslinked copolymer of monovinyl aromatic monomer, monovinyl aliphatic monomer, and polyvinyl aromatic monomer; chromatography THE DOW CHEMICAL COMPANY (US) 1995-10-24 US disclosed
US-5185157-A With solid or liquid carrier, free of zinc, magnesium and calcium salts TYSON & ASSOCIATES, INC. 1993-02-09 US disclosed
US-4778808-A CONCENTRATING CULTURE BROTH WHILE CONTROLLING PH AND TEMPERATURE STABILITY AJINOMOTO CO., INC. (JP) 1988-10-18 US disclosed