SCHEMBL22301396

SCHEMBL22301396

NNc1cc(Cl)nc(Cl)c1N

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.32
HTT P42858 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2767477 0.81 KMT2A (0.35) KMT2AMEN1HTTTDP1CYP2D6
SCHEMBL31248906 0.81 KMT2A (0.35) KMT2AMEN1HTTTDP1CYP2D6
SCHEMBL5067867 0.76 KDM4E (0.36) KMT2AHTTCYP2D6CYP2C19ALDH1A1
SCHEMBL31426069 0.76 KDM4E (0.36) KMT2AHTTCYP2D6CYP2C19ALDH1A1
SCHEMBL15817308 0.75 S1PR2 (0.40) KMT2AMEN1HTTTDP1CYP2D6
SCHEMBL9476338 0.74 ALDH1A1 (0.46) KMT2AMEN1HTTTDP1ALDH1A1
SCHEMBL29462391 0.72 TDP1 (0.48) KMT2AMEN1HTTTDP1CYP2D6
SCHEMBL259983 0.72 TDP1 (0.48) KMT2AMEN1HTTTDP1CYP2D6
Hydrochloric Acid SCHEMBL5778836 0.70 TDP1 (0.46) KMT2AMEN1HTTTDP1ALDH1A1
SCHEMBL23137233 0.70 ALDH1A1 (0.33) KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020159905-A1 PYRAZOLOPYRIDINES AND TRIAZOLOPYRIDINES AS A2A / A2B INHIBITORS INCYTE CORPORATION (US) 2020-08-06 WO disclosed