SCHEMBL259983

SCHEMBL259983

Nc1cc(Cl)nc(Cl)c1N

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
KMT2A Q03164 4/20 0.37
MEN1 O00255 2/20 0.37
HTT P42858 1/20 0.37
GAA P10253 1/20 0.35
HSP90AB1 P08238 4/20 0.33
HSP90AA1 P07900 3/20 0.33
KDM4E B2RXH2 2/20 0.33
CDK2 P24941 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29462391 1.00 TDP1 (0.48) TDP1KMT2AMEN1HTTGAA
Hydrochloric Acid SCHEMBL5778836 0.97 TDP1 (0.46) TDP1KMT2AMEN1HTTGAA
SCHEMBL9476338 0.81 ALDH1A1 (0.46) TDP1KMT2AMEN1HTTGAA
SCHEMBL38657291 0.79 TDP1 (0.48) TDP1KMT2AMEN1GAAHSP90AB1
SCHEMBL26694654 0.79 TDP1 (0.48) TDP1KMT2AMEN1GAAHSP90AB1
SCHEMBL25292365 0.75 GAA (0.40) TDP1KMT2AMEN1HTTGAA
SCHEMBL5746102 0.75 ALDH1A1 (0.40) TDP1KMT2AMEN1HTTGAA
SCHEMBL19049647 0.75 TDP1 (0.44) TDP1KMT2AGAAHSP90AB1HSP90AA1
SCHEMBL18260463 0.75 TDP1 (0.44) TDP1KMT2AMEN1GAAHSP90AB1
SCHEMBL30421541 0.75 ALDH1A1 (0.40) TDP1KMT2AMEN1HTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 206 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078127-A1 HETEROBICYCLIC AMIDES AS INHIBITORS OF CD38 BOEHRINGER INGELHEIM INT (DE) 2026-03-19 US disclosed
US-20250325544-A1 CDK INHIBITORS GENENTECH, INC. (US) 2025-10-23 US disclosed
US-12428425-B2 Heterocyclic compounds as triggering receptor expressed on myeloid cells 2 agonists and methods of use AMGEN INC. (US) 2025-09-30 US disclosed
US-20250281487-A1 CDK INHIBITORS GENENTECH, INC. (US) 2025-09-11 US disclosed
US-20250275971-A1 CDK INHIBITORS GENENTECH, INC. (US) 2025-09-04 US disclosed
US-20250275972-A1 CDK INHIBITORS GENENTECH, INC. (US) 2025-09-04 US disclosed
US-12398146-B2 Heterobicyclic amides as inhibitors of CD38 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2025-08-26 US disclosed
US-12285429-B2 CDK inhibitors GENENTECH, INC. (US) 2025-04-29 US disclosed
EP-4524135-A1 KINESIN KIF18A INHIBITOR AND USE THEREOF Shanghai Apeiron Therapeutics Company Limited (CN) 2025-03-19 EP disclosed
US-20250064806-A1 CDK INHIBITORS GENENTECH, INC. 2025-02-27 US disclosed
WO-1995018616-A2 8-AZA, 6-AZA AND 6,8-DIAZA-1,4-DIHYDROQUINOXALINE-2,3-DIONES AND THE USE THEREOF AS ANTAGONISTS FOR THE GLYCINE/NMDA RECEPTOR ACEA PHARM INC (US) 1995-07-13 WO disclosed
EP-0505893-A1 Imidazopyridines MERCK PATENT GmbH (DE) 1992-09-30 EP disclosed
EP-0255217-B1 FUSED IMIDAZOHETEROCYCLIC COMPOUNDS A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1992-01-22 EP disclosed
US-4948800-A MUSCLE RELAXANTS; ANTICONVULSANTS; ANXIOLYTIC AGENTS; 3-HYDROXYALKYL-PYRIDO(4,5-B OR-C)IMIDAZOLE COMPOUNDS A. H. ROBINS COMPANY, INCORPORATED (US) 1990-08-14 US disclosed
US-4914109-A ANTICONVULSANTS, ANTIANXIETY AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1990-04-03 US disclosed
US-4873251-A MUSCLE RELAXANTS, ANTICONVULSANTS, ANTIANXIETY AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1989-10-10 US disclosed
US-4824951-A MUSCLE RELAXANTS, ANTICONVULSANTS, ANXIOLYTIC AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1989-04-25 US disclosed
US-4772600-A MUSCLE RELAXANTS, ANTICONVULSANTS, ANXIOLYTIC A. H. ROBINS COMPANY, INC. (US) 1988-09-20 US disclosed
EP-0255217-A1 Fused imidazoheterocyclic compounds A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1988-02-03 EP disclosed
US-3935195-A FLUORESCENT DYE STERLING DRUG INC. (US) 1976-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12428425-B2 Heterocyclic compounds as triggering receptor expressed on myeloid cells 2 agonists and methods of use MSR1, FPR2, CD14 TDP1 697/4885KMT2A 1950/4885MEN1 3486/4885
US-20250281487-A1 CDK INHIBITORS CDK6, CDK9, CDKL1 TDP1 968/4885KMT2A 178/4885MEN1 1620/4885
US-20250064806-A1 CDK INHIBITORS CDK9, CDK6, CDK3 TDP1 1013/4885KMT2A 147/4885MEN1 2306/4885
US-12285429-B2 CDK inhibitors CDK9, CDK3, CDKL1 TDP1 844/4885KMT2A 151/4885MEN1 1846/4885
US-12398146-B2 Heterobicyclic amides as inhibitors of CD38 CD38, PARP12, ENTPD2 TDP1 1007/4885KMT2A 1094/4885MEN1 3571/4885
US-20260078127-A1 HETEROBICYCLIC AMIDES AS INHIBITORS OF CD38 CD38, CD22, CD79B TDP1 2127/4885KMT2A 2514/4885MEN1 4829/4885
US-20250325544-A1 CDK INHIBITORS CDK6, CDK9, CDKL1 TDP1 968/4885KMT2A 178/4885MEN1 1620/4885
US-20250275972-A1 CDK INHIBITORS CDK9, CDK6, CDK3 TDP1 1013/4885KMT2A 147/4885MEN1 2306/4885
US-20250275971-A1 CDK INHIBITORS CDK6, CDK9, CDKL1 TDP1 968/4885KMT2A 178/4885MEN1 1620/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.