SCHEMBL22322112

SCHEMBL22322112

[CH2]COc1ccc(C=O)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.52
TTR P02766 1/20 0.46
MAPT P10636 3/20 0.46
HPGD P15428 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
FDPS P14324 1/20 0.45
LMNA P02545 2/20 0.44
TSHR P16473 1/20 0.43
TACR2 P21452 1/20 0.42
ALDH1A3 P47895 2/20 0.41
ALDH3A1 P30838 1/20 0.41
NPC1 O15118 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL944430 0.83 ALDH1A1 (0.48) ALDH1A1TTRMAPTHPGDCYP1A2
SCHEMBL566725 0.82 ALDH1A1 (0.60) ALDH1A1TTRMAPTHPGDCYP1A2
SCHEMBL30902399 0.82 ALDH1A1 (0.60) ALDH1A1TTRMAPTHPGDCYP1A2
SCHEMBL29956255 0.81 ALDH1A1 (0.47) ALDH1A1TTRMAPTHPGDCYP1A2
SCHEMBL566342 0.79 CSNK2A1 (0.55) ALDH1A1MAPTHPGDCYP1A2CYP2D6
Benzene SCHEMBL27642249 0.79 TACR2 (0.57) ALDH1A1MAPTHPGDCYP1A2CYP2D6
SCHEMBL31474820 0.79 ALDH1A1 (0.50) ALDH1A1TTRMAPTHPGDCYP1A2
SCHEMBL31471675 0.79 ALDH1A1 (0.50) ALDH1A1TTRMAPTHPGDCYP1A2
SCHEMBL2560176 0.79 ALDH1A1 (0.44) ALDH1A1TTRMAPTHPGDCYP1A2
SCHEMBL22322051 0.79 FDPS (0.49) ALDH1A1MAPTHPGDFDPSLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3921320-A1 IMIDAZO [2, 1-F] [1, 2, 4] TRIAZIN-4-AMINE DERIVATIVES AS TLR7 AGONIST BeiGene, Ltd. (KY) 2021-12-15 EP disclosed
CN-113454086-A Imidazo [2,1-F ] [1,2,4] triazin-4-amine derivatives as TLR7 agonists 百济神州有限公司 2021-09-28 CN disclosed
WO-2020160711-A1 IMIDAZO [2, 1-F] [1, 2, 4] TRIAZIN-4-AMINE DERIVATIVES AS TLR7 AGONIST BEIGENE, LTD. (KY) 2020-08-13 WO disclosed