SCHEMBL2232838

SCHEMBL2232838

CCOC(=O)/C=C/c1cc(C)c(Oc2ccc(O)cn2)c(C)c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA7 P43166 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
CYP3A4 P08684 2/20 0.49
TTR P02766 1/20 0.48
DPP4 P27487 1/20 0.48
ESR1 P03372 4/20 0.46
FDPS P14324 1/20 0.46
MAOB P27338 1/20 0.44
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PTGS2 P35354 1/20 0.41
MET P08581 2/20 0.40
BCHE P06276 2/20 0.39
ACHE P22303 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13582495 0.85 ESR1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL13582500 0.85 ESR1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL2232047 0.84 APP (0.47) CA12CA1CA2CA7CA9
SCHEMBL2232050 0.84 APP (0.47) CA12CA1CA2CA7CA9
SCHEMBL2298327 0.80 CA12 (0.38) CA12CA1CA2CA7CA9
SCHEMBL2231437 0.80 CA12 (0.38) CA12CA1CA2CA7CA9
SCHEMBL13582160 0.78 ESR1 (0.38) CA12CA1CA2CA7CA9
SCHEMBL13582158 0.78 ESR1 (0.38) CA12CA1CA2CA7CA9
SCHEMBL2234037 0.77 GPR183 (0.42)
SCHEMBL2301371 0.77 REN (0.41) ESR1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed