SCHEMBL2298327

SCHEMBL2298327

CCOC(=O)/C=C/c1cc(C)c(Oc2ccc(OCc3cscn3)cn2)c(C)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CYP3A4 P08684 2/20 0.38
FDPS P14324 1/20 0.37
ESR1 P03372 5/20 0.37
TTR P02766 1/20 0.36
DPP4 P27487 1/20 0.36
MAOB P27338 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ACHE P22303 4/20 0.34
BCHE P06276 3/20 0.34
PTGS2 P35354 1/20 0.34
BACE1 P56817 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13582005 0.90 CYP4F2 (0.36) CA2CA9ESR1
SCHEMBL13582003 0.90 CYP4F2 (0.36) CA2CA9ESR1
SCHEMBL2231437 0.84 CA12 (0.38) CA12CA1CA2CA7CA9
SCHEMBL2298336 0.82 ESR1 (0.36) ESR1BACE1
SCHEMBL2232838 0.80 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL2298330 0.78 MAPK14 (0.34)
SCHEMBL2235396 0.75 GPR183 (0.45) ACHE
SCHEMBL2235620 0.75 GPR183 (0.41) MAOBACHEBCHE
SCHEMBL2235390 0.75 GPR183 (0.45) ACHE
Hydrochloric Acid SCHEMBL13583010 0.74 GPR183 (0.45) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed