SCHEMBL22330601

SCHEMBL22330601

CCOc1ccc(-c2cc(C)c(C)n2-c2ccc(S(N)(=O)=O)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 11/20 0.64
PTGS2 P35354 6/20 0.57
CA1 P00915 2/20 0.57
CA2 P00918 2/20 0.57
PTGS1 P23219 2/20 0.57
CA12 O43570 1/20 0.57
CA7 P43166 1/20 0.57
CA9 Q16790 1/20 0.57
CYP2D6 P10635 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21675742 0.89 CHRNA7 (0.58) CHRNA7PTGS2CA1CA2PTGS1
Apricoxib SCHEMBL3435344 0.81 CA1 (0.60) CHRNA7PTGS2CA1CA2PTGS1
Apricoxib SCHEMBL346028 0.81 CA1 (0.60) CHRNA7PTGS2CA1CA2PTGS1
SCHEMBL2464617 0.80 PTGS2 (0.59) CHRNA7PTGS2CA1CA2PTGS1
SCHEMBL3031000 0.77 CHRNA7 (0.98) CHRNA7CA12CA9CYP2D6
SCHEMBL5312990 0.77 CHRNA7 (0.60) CHRNA7PTGS2CA1CA2PTGS1
SCHEMBL2841663 0.76 PTGS2 (0.60) CHRNA7PTGS2CA1CA2PTGS1
SCHEMBL5308912 0.76 PTGS2 (0.64) PTGS2CA1CA2PTGS1CA12
SCHEMBL17920087 0.76 PTGS2 (0.64) PTGS2CA1CA2PTGS1CA12
SCHEMBL4706398 0.76 CA2 (1.00) PTGS2CA1CA2PTGS1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3693022-A2 COX-2-TARGETING, PLATINUM-CONTAINING CONJUGATES AND THEIR USE IN THE TREATMENT OF TUMORS AND CANCERS Reiley Pharmaceuticals, Inc. (US) 2020-08-12 EP disclosed