SCHEMBL2233135

SCHEMBL2233135

CCCCOC(=O)/C=C/c1ccc(Oc2ccc(O)cn2)cc1C

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.48
APP P05067 5/20 0.45
AKR1B10 O60218 6/20 0.42
AKR1B1 P15121 6/20 0.42
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2230602 0.85 MAPT (0.44) ESR1APP
SCHEMBL13581749 0.82 ESR1 (0.52) ESR1
SCHEMBL2354427 0.82 ESR1 (0.52) ESR1
SCHEMBL28368058 0.79 APP (0.52) ESR1APPAKR1B10AKR1B1ATM
SCHEMBL27463292 0.79 APP (0.52) ESR1APPAKR1B10AKR1B1ATM
SCHEMBL9820613 0.79 APP (0.57) ESR1APPAKR1B10AKR1B1
SCHEMBL2232050 0.79 APP (0.47) ESR1APPAKR1B10AKR1B1
SCHEMBL2232047 0.79 APP (0.47) ESR1APPAKR1B10AKR1B1
SCHEMBL2233144 0.78 ALOX5 (0.47)
SCHEMBL14289647 0.78 ESR1 (0.56) ESR1APPATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed