SCHEMBL2233272

SCHEMBL2233272

Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ccc(C(F)(F)F)cc3)C2c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 8/20 0.52
RXFP1 Q9HBX9 3/20 0.50
ANXA2 P07355 3/20 0.48
S100A10 P60903 3/20 0.48
CCR2 P41597 3/20 0.47
KDM4E B2RXH2 3/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
HPGD P15428 2/20 0.43
P2RX3 P56373 2/20 0.41
LMNA P02545 1/20 0.41
ATM Q13315 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2301658 0.93 CCR1 (0.54) CCR1RXFP1ANXA2S100A10CCR2
SCHEMBL2233975 0.91 ANXA2 (0.49) CCR1RXFP1ANXA2S100A10CCR2
SCHEMBL2232399 0.85 CCR1 (0.54) CCR1RXFP1ANXA2S100A10CCR2
SCHEMBL2235286 0.81 ANXA2 (0.67) CCR1ANXA2S100A10MEN1KMT2A
SCHEMBL10116868 0.80 KDM4E (0.65) CCR1RXFP1CCR2KDM4EMEN1
SCHEMBL10116779 0.78 P2RX3 (0.56) CCR1RXFP1CCR2KDM4EMEN1
SCHEMBL10116809 0.77 RXFP1 (0.69) CCR1RXFP1KDM4EMEN1KMT2A
SCHEMBL10117163 0.77 P2RX3 (0.59) CCR1RXFP1KDM4EMEN1KMT2A
SCHEMBL6116461 0.77 RXFP1 (0.48) CCR1RXFP1ANXA2S100A10CCR2
SCHEMBL10146036 0.76 RXFP1 (0.69) CCR1RXFP1CCR2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO claimed
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO disclosed