SCHEMBL2301658

SCHEMBL2301658

Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccc3)C2c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 7/20 0.54
ANXA2 P07355 2/20 0.50
S100A10 P60903 2/20 0.50
RXFP1 Q9HBX9 3/20 0.49
KDM4E B2RXH2 3/20 0.47
HPGD P15428 3/20 0.47
P2RX3 P56373 3/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
LMNA P02545 1/20 0.45
CCR2 P41597 2/20 0.44
HIF1A Q16665 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2233272 0.93 CCR1 (0.52) CCR1ANXA2S100A10RXFP1KDM4E
SCHEMBL2233975 0.88 ANXA2 (0.49) CCR1ANXA2S100A10RXFP1KDM4E
SCHEMBL10146036 0.80 RXFP1 (0.69) CCR1RXFP1KDM4EHPGDP2RX3
SCHEMBL2235286 0.80 ANXA2 (0.67) CCR1ANXA2S100A10MEN1KMT2A
SCHEMBL10116868 0.79 KDM4E (0.65) CCR1RXFP1KDM4EHPGDP2RX3
SCHEMBL2232399 0.78 CCR1 (0.54) CCR1ANXA2S100A10RXFP1KDM4E
SCHEMBL2232358 0.78 CCR1 (0.59) CCR1ANXA2S100A10RXFP1KDM4E
SCHEMBL10116779 0.77 P2RX3 (0.56) CCR1RXFP1KDM4EHPGDP2RX3
SCHEMBL10120635 0.76 CCR1 (0.69) CCR1RXFP1KDM4EHPGDP2RX3
SCHEMBL10120633 0.76 CCR1 (0.65) CCR1RXFP1KDM4EHPGDP2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO disclosed