SCHEMBL22336875

SCHEMBL22336875

COCCOc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCO

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.87
ERBB2 P04626 4/20 0.73
HDAC3 O15379 3/20 0.73
HDAC4 P56524 3/20 0.73
HDAC1 Q13547 3/20 0.73
HDAC7 Q8WUI4 3/20 0.73
HDAC2 Q92769 3/20 0.73
HDAC10 Q969S8 3/20 0.73
HDAC11 Q96DB2 3/20 0.73
HDAC8 Q9BY41 3/20 0.73
HDAC6 Q9UBN7 3/20 0.73
HDAC9 Q9UKV0 3/20 0.73
HDAC5 Q9UQL6 3/20 0.73
FBP1 P09467 2/20 0.71
AURKA O14965 1/20 0.70
INSR P06213 1/20 0.70
PDGFRB P09619 1/20 0.70
FLT4 P35916 1/20 0.70
KDR P35968 1/20 0.70
CLK1 P49759 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22338174 0.95 EGFR (0.80) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL15217656 0.94 EGFR (0.90) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL1730545 0.93 EGFR (1.00) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL24535320 0.89 EGFR (0.72) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL25083284 0.89 EGFR (0.71) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL18978997 0.87 EGFR (0.89) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL8211574 0.87 HDAC3 (0.89) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL10118455 0.87 HDAC3 (0.83) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL6994526 0.87 EGFR (0.69) EGFRERBB2HDAC3HDAC4HDAC1
SCHEMBL4343029 0.87 EGFR (0.87) EGFRERBB2HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020163598-A1 IMMUNOPHILIN-DEPENDENT INHIBITORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-08-13 WO disclosed