SCHEMBL22337945

SCHEMBL22337945

CNc1ccnc2ccoc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.34
UTS2R Q9UKP6 1/20 0.33
IKBKE Q14164 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
CDC42BPA Q5VT25 1/20 0.33
CDC42BPB Q9Y5S2 1/20 0.33
NR4A2 P43354 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTR1A P08908 3/20 0.32
ADRA1D P25100 3/20 0.32
ADRA1A P35348 3/20 0.32
ADRA1B P35368 3/20 0.32
ASIC3 Q9UHC3 1/20 0.31
AURKA O14965 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20265612 0.80 IKBKE (0.33) IRAK4UTS2RIKBKETBK1HTR1A
SCHEMBL13454732 0.72 CCR1 (0.38) IRAK4CYP1A2HSD17B10ASIC3
SCHEMBL20778909 0.71 MTNR1A (0.42) HSD17B10
SCHEMBL30748895 0.71 IRAK4 (0.52) IRAK4CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL29487180 0.68 NR4A2 (0.34) IRAK4NR4A2CYP1A2CYP2C9CYP2C19
SCHEMBL13262134 0.68 NCF1 (0.43) IRAK4NR4A2
SCHEMBL15339587 0.68 PRKCI (0.32) IRAK4
SCHEMBL30504301 0.68 NCF1 (0.43) IRAK4NR4A2
SCHEMBL2798723 0.68 NR4A2 (0.34) IRAK4NR4A2CYP1A2CYP2C9CYP2C19
SCHEMBL29446635 0.68 IRAK4 (0.30) IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020163193-A1 BICYCLIC ETHER O-GLYCOPROTEIN-2-ACETAMIDO-2-DEOXY-3-D-GLUCOPYRANOSIDASE INHIBITORS BIOGEN MA INC. (US) 2020-08-13 WO disclosed