Prednisolone

Prednisolone

SCHEMBL2233875

C[C@]12C=CC(=O)C=C1CCC1C2C(O)C[C@@]2(C)C1CC[C@]2(O)C(=O)CO.O=P([O-])([O-])[O-].[Na+].[Na+].[Na+]

nearest known ligand 0.90

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Prednisolone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 10/20 0.90
HIF1A Q16665 9/20 0.90
HSD17B10 Q99714 8/20 0.90
PGR P06401 5/20 0.90
CYP3A4 P08684 4/20 0.90
CYP2C19 P33261 3/20 0.90
ABCB11 O95342 2/20 0.90
SERPINA6 P08185 2/20 0.90
NR3C2 P08235 2/20 0.90
TNF P01375 1/20 0.90
IL6 P05231 1/20 0.90
AR P10275 1/20 0.90
GLUL P15104 1/20 0.90
ADAM17 P78536 1/20 0.90
GPBAR1 Q8TDU6 1/20 0.90
LMNA P02545 2/20 0.69
ALDH1A1 P00352 2/20 0.64
ABCC4 O15439 1/20 0.64
NR1I2 O75469 1/20 0.64
PDE4D Q08499 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prednisolone SCHEMBL23564 1.00 NR3C1 (0.90) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL4751186 0.97 NR3C1 (0.85) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL1930093 0.97 NR3C1 (0.88) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL7514 0.95 NR3C1 (0.93) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL16094487 0.95 NR3C1 (0.93) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL5504548 0.95 NR3C1 (0.93) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL23863778 0.95 NR3C1 (1.00) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL13044469 0.95 NR3C1 (1.00) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL2737385 0.95 NR3C1 (1.00) NR3C1HIF1AHSD17B10PGRCYP3A4
Prednisolone SCHEMBL765329 0.95 NR3C1 (1.00) NR3C1HIF1AHSD17B10PGRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117337297-A Use of SOS1 inhibitors and MTOR inhibitors for the treatment of cancer 锐新医药公司 2024-01-02 CN disclosed
US-20230041980-A1 METHOD OF PROTECTING A RESPIRATORY TRACT OR A LUNG FROM DAMAGE, METHOD OF PROTECTING A LUNG FROM PRESSURE DAMAGE INDUCED BY A VENTILATOR, METHOD OF SUPPRESSING SPREAD OF INFECTION WITH VIRUSES OR BACTERIA THAT CAUSE PNEUMONIA IN PULMONARY BRONCHIAL EPITHELIAL CELLS OR ALVEOLAR EPITHELIAL CELLS, AND NASAL SPRAY NEXT21 KABUSHIKI KAISHA (JP) 2023-02-09 US disclosed
EP-4125927-A1 MEDICINE CONTAINING TREHALOSE OR TREHALOSE DERIVATIVE AND NASAL SPRAY Next21 Kabushiki Kaisha (JP) 2023-02-08 EP disclosed
WO-2021210648-A1 MEDICINE CONTAINING TREHALOSE OR TREHALOSE DERIVATIVE AND NASAL SPRAY NEXT21 KABUSHIKI KAISHA (JP) 2021-10-21 WO disclosed
WO-2021025140-A1 DUAL-SPECIFIC PROTEIN 小野薬品工業株式会社 2021-02-11 WO disclosed
WO-2021020416-A1 BISPECIFIC ANTIBODY 小野薬品工業株式会社 2021-02-04 WO disclosed
WO-2019172419-A1 METHOD FOR DETECTING INDICATOR OF IMMUNE-RELATED DISEASE 株式会社マンダム 2019-09-12 WO disclosed
WO-2019163838-A1 MARKER FOR MULTIPLE SCLEROSIS 国立研究開発法人理化学研究所 2019-08-29 WO disclosed
WO-2019156199-A1 BISPECIFIC ANTIBODY 小野薬品工業株式会社 2019-08-15 WO disclosed
EP-2353592-A1 Therapeutic causing contraction of mucosal tissue and method of treating diseases relating to mucosal tissues Japan Science and Technology Agency (JP) 2011-08-10 EP disclosed
US-20050187303-A1 Therapeutic causing contraction of mucosal tissue, method of treating diseases relating to mucosal tissues, injector and therapeutic set JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2005-08-25 US disclosed
EP-1557163-A1 THERAPEUTIC CAUSING CONTRACTION OF MUCOSAL TISSUE, METHOD OF TREATING DISEASES RELATING TO MUCOSAL TISSUES, INJECTOR AND THERAPEUTIC SET Japan Science and Technology Agency (JP) 2005-07-27 EP disclosed
EP-1197209-A1 PERCUTANEOUSLY ABSORBABLE PREPARATIONS HISAMITSU PHARMACEUTICAL CO. INC. (JP) 2002-04-17 EP disclosed
EP-1190706-A1 LIPOSOMES TERUMO KABUSHIKI KAISHA (JP) 2002-03-27 EP disclosed
EP-0953357-A1 NEPHROTROPIC DRUGS Drug Delivery System Institute, Ltd. (JP) 1999-11-03 EP disclosed
EP-0308572-B1 An iontophoresis device HISAMITSU PHARMACEUTICAL CO (JP) 1995-11-08 EP disclosed
EP-0138347-B1 AN IONTOPHORESIS DEVICE KABUSHIKI KAISYA ADVANCE (JP) 1989-08-02 EP disclosed
EP-0308572-A2 An iontophoresis device Hisamitsu Pharmaceutical Co., Inc. (JP) 1989-03-29 EP disclosed
US-4764164-A Iontophoresis device KABUSHIKI KAISYA ADVANCE KAIHATSU KENKYUJO (JP) 1988-08-16 US disclosed
EP-0138347-A1 An iontophoresis device KABUSHIKI KAISYA ADVANCE (JP) 1985-04-24 EP disclosed