SCHEMBL22341925

SCHEMBL22341925

COc1c(C)c(Br)cc(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.39
CA4 P22748 2/20 0.39
ACHE P22303 1/20 0.32
IMPDH2 P12268 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
TUBB1 Q9H4B7 1/20 0.31
TPMT P51580 1/20 0.31
TSHR P16473 1/20 0.30
APOBEC3A P31941 1/20 0.30
HTT P42858 1/20 0.30
APOBEC3G Q9HC16 1/20 0.30
CA1 P00915 1/20 0.30
CA6 P23280 1/20 0.30
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27628106 0.83 CA2 (0.43) CA2CA4ACHEALOX5APFEN1
SCHEMBL27628234 0.83 CA2 (0.39) CA2CA4ACHEIMPDH2ALOX5AP
SCHEMBL31015964 0.83 CA2 (0.41) CA2CA4ALOX5APFEN1HSD17B10
SCHEMBL9377977 0.83 CA2 (0.41) CA2CA4ALOX5APFEN1HSD17B10
SCHEMBL16256381 0.80 ACHE (0.36) ACHEALDH1A1TUBB1
SCHEMBL4589673 0.78 CA2 (0.46) CA2CA4ALOX5APFEN1HSD17B10
SCHEMBL9549445 0.78 CA2 (0.38) CA2CA4ALOX5APFEN1HSD17B10
SCHEMBL22831899 0.78 MAPT (0.38) CA2CA4ALOX5APFEN1HSD17B10
SCHEMBL525151 0.77 CA2 (0.50) CA2CA4ACHEIMPDH2ALOX5AP
SCHEMBL15510333 0.76 CA2 (0.36) CA2CA4ACHEIMPDH2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3484878-B1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2020-08-19 EP disclosed