SCHEMBL22341998

SCHEMBL22341998

CC(C)(O)CNC(=O)c1ccc(NC(=O)O)cn1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 7/20 0.48
ADORA2A P29274 1/20 0.45
HDAC3 O15379 3/20 0.45
HDAC4 P56524 3/20 0.45
HDAC1 Q13547 3/20 0.45
HDAC8 Q9BY41 3/20 0.45
HDAC6 Q9UBN7 3/20 0.45
EGLN1 Q9GZT9 1/20 0.44
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CNR2 P34972 1/20 0.42
NAMPT P43490 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22341957 0.88 CNR2 (0.48) P4HTMADORA2AHDAC3HDAC4HDAC1
SCHEMBL22341942 0.86 P4HTM (0.46) P4HTMADORA2AHDAC3HDAC4HDAC1
SCHEMBL28940895 0.83 P4HTM (0.41) P4HTMADORA2AHDAC3HDAC4HDAC1
SCHEMBL28940979 0.82 CNR2 (0.38) P4HTMNPC1ALDH1A1GAARAB9A
SCHEMBL21379406 0.81 NAMPT (0.48) P4HTMHDAC3HDAC4HDAC1HDAC8
SCHEMBL28292587 0.79 HDAC3 (0.47) P4HTMHDAC3HDAC4HDAC1HDAC8
SCHEMBL22341853 0.79 ANO1 (0.50)
SCHEMBL22227949 0.79 P4HTM (0.55) P4HTMHDAC3HDAC4HDAC1HDAC8
SCHEMBL30064984 0.78 KDM4E (0.50) EGLN1ALDH1A1CNR2
SCHEMBL29085188 0.78 KDM4E (0.50) EGLN1ALDH1A1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
EP-3484878-B1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2020-08-19 EP claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed