SCHEMBL28292587

SCHEMBL28292587

CC(O)CNC(=O)c1ccc(NC(=O)O)cn1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 7/20 0.47
HDAC1 Q13547 7/20 0.47
HDAC8 Q9BY41 7/20 0.47
HDAC4 P56524 4/20 0.47
HDAC6 Q9UBN7 4/20 0.47
P4HTM Q9NXG6 7/20 0.47
NAMPT P43490 2/20 0.46
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 2/20 0.43
EGLN1 Q9GZT9 1/20 0.43
MAPT P10636 1/20 0.43
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28940920 0.81 ACR (0.40) P4HTMNAMPTSMN1; SMN2ALDH1A1
SCHEMBL21379406 0.80 NAMPT (0.48) HDAC3HDAC1HDAC8HDAC4HDAC6
SCHEMBL21379443 0.80 ANO1 (0.46)
SCHEMBL21379445 0.80 ANO1 (0.46)
SCHEMBL22341998 0.79 P4HTM (0.48) HDAC3HDAC1HDAC8HDAC4HDAC6
SCHEMBL20929477 0.78 ADORA2A (0.44)
SCHEMBL25745885 0.78 NAMPT (0.48) HDAC3HDAC1HDAC8HDAC4HDAC6
SCHEMBL22227949 0.77 P4HTM (0.55) HDAC3HDAC1HDAC8HDAC4HDAC6
SCHEMBL12789191 0.77 EGLN1 (0.52) HDAC3HDAC1HDAC6P4HTMNPC1
SCHEMBL22341942 0.77 P4HTM (0.46) HDAC3HDAC1HDAC8HDAC4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed