SCHEMBL22345944

SCHEMBL22345944

CN(C)[C@@H](Cc1cn(C)c2ccccc12)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.51
KDM4E B2RXH2 4/20 0.49
CMA1 P23946 2/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
RECQL P46063 1/20 0.47
CA2 P00918 1/20 0.47
ADAM17 P78536 1/20 0.47
HTR2A P28223 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
LMNA P02545 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3304505 1.00 GPR84 (0.51) GPR84KDM4ECMA1HPGDHSD17B10
Ammonia Solution, Strong SCHEMBL27663008 0.99 GPR84 (0.50) GPR84KDM4ECMA1HPGDHSD17B10
SCHEMBL28406976 0.99 GPR84 (0.50) GPR84KDM4ECMA1HPGDHSD17B10
Iodide SCHEMBL28079826 0.97 GPR84 (0.49) GPR84KDM4ECMA1HPGDHSD17B10
Hydrochloric Acid SCHEMBL27640400 0.97 GPR84 (0.49) GPR84KDM4ECMA1HPGDHSD17B10
SCHEMBL27693089 0.84 ALDH1A1 (0.48) ALDH1A1MAPTRECQLCA2MEN1
SCHEMBL4297919 0.82 HDAC3 (0.44) GPR84KDM4ECMA1HPGDHSD17B10
SCHEMBL25469062 0.81 GPR84 (0.56) GPR84KDM4ECMA1HPGDHSD17B10
SCHEMBL9275407 0.81 GPR84 (0.56) GPR84KDM4ECMA1HPGDHSD17B10
SCHEMBL18413853 0.81 GPR84 (0.56) GPR84KDM4ECMA1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020166592-A1 HEMIASTERLIN DERIVATIVE AND ANTIBODY-DRUG CONJUGATE THEREOF 大日本住友製薬株式会社 2020-08-20 WO disclosed
WO-2020166600-A1 HEMIASTERLIN DERIVATIVE HAVING CYSTEINE RESIDUE 大日本住友製薬株式会社 2020-08-20 WO disclosed