SCHEMBL22345951

SCHEMBL22345951

CC(C)(C)OC(=O)N[C@H](C(=O)OC(C)(C)C)C(C)(C)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 9/20 0.48
CTSK P43235 8/20 0.48
CTSB P07858 2/20 0.46
CTSL P07711 1/20 0.46
ATM Q13315 1/20 0.45
PPARA Q07869 3/20 0.42
PPARG P37231 2/20 0.42
SYK P43405 1/20 0.42
ACE P12821 1/20 0.41
KLK5 Q9Y337 1/20 0.41
PPARD Q03181 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL58075 0.93 CTSS (0.47) CTSSCTSKCTSBCTSLATM
SCHEMBL89265 0.93 CTSS (0.47) CTSSCTSKCTSBCTSLATM
SCHEMBL5024738 0.89 CTSS (0.49) CTSSCTSKCTSBCTSLATM
SCHEMBL58394 0.89 CTSS (0.49) CTSSCTSKCTSBCTSLATM
SCHEMBL57550 0.89 CTSS (0.49) CTSSCTSKCTSBCTSLATM
SCHEMBL6671005 0.87 CTSS (0.47) CTSSCTSKCTSBCTSLATM
SCHEMBL9963924 0.81 CTSS (0.52) CTSSCTSKCTSBCTSLATM
SCHEMBL18405913 0.81 CTSS (0.52) CTSSCTSKCTSBCTSLATM
SCHEMBL18932855 0.81 PPARA (0.43) CTSSCTSKCTSBCTSLATM
SCHEMBL18932852 0.80 PPARA (0.42) CTSSCTSKCTSBCTSLATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020166592-A1 HEMIASTERLIN DERIVATIVE AND ANTIBODY-DRUG CONJUGATE THEREOF 大日本住友製薬株式会社 2020-08-20 WO disclosed
WO-2020166600-A1 HEMIASTERLIN DERIVATIVE HAVING CYSTEINE RESIDUE 大日本住友製薬株式会社 2020-08-20 WO disclosed