SCHEMBL22352873

SCHEMBL22352873

N#CC12CCC(CNc3cccc(Br)c3)(CC1)C2

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
GAA P10253 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAPT P10636 1/20 0.36
PRKCQ Q04759 2/20 0.35
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HTT P42858 1/20 0.32
MAP2K1 Q02750 1/20 0.32
GRK2 P25098 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22347387 0.92 ALDH1A1 (0.37) ALDH1A1GAAL3MBTL1MAPTPRKCQ
SCHEMBL22353922 0.76 GAA (0.40) ALDH1A1GAAL3MBTL1DRD4DRD3
SCHEMBL22352872 0.73 PRKCQ (0.38) ALDH1A1GAAL3MBTL1MAPTPRKCQ
SCHEMBL22353831 0.73 PRKCQ (0.36) ALDH1A1GAAL3MBTL1MAPTPRKCQ
SCHEMBL22347208 0.71
SCHEMBL22347580 0.71 GAA (0.46) ALDH1A1GAAL3MBTL1MAPTSMN1; SMN2
SCHEMBL31608504 0.71 GAA (0.46) ALDH1A1GAAL3MBTL1MAPTSMN1; SMN2
SCHEMBL22347657 0.70 GAA (0.41) ALDH1A1GAAL3MBTL1SMN1; SMN2HTT
SCHEMBL22347206 0.70 HTR1A (0.36) ALDH1A1GAAL3MBTL1DRD4DRD3
SCHEMBL22347929 0.70 IDO1 (0.35) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020168148-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-08-20 WO disclosed