SCHEMBL22354072

SCHEMBL22354072

C=C(F)CCC(=O)N(CCCCCc1nnc(C2CC2)o1)c1cccc(Br)c1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.34
LMNA P02545 2/20 0.34
ALDH1A1 P00352 5/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
NPC1 O15118 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NR1H4 Q96RI1 6/20 0.33
GAA P10253 1/20 0.32
TP53 P04637 1/20 0.31
GPX4 P36969 1/20 0.31
PAX8 Q06710 1/20 0.31
TNKS O95271 1/20 0.30
PARP1 P09874 1/20 0.30
PARP2 Q9UGN5 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24259062 0.86 ALDH1A1 (0.35) RAB9ALMNAALDH1A1HTTKMT2A
SCHEMBL24258760 0.83 AKR1C4 (0.36) L3MBTL1NR1H4MAPT
SCHEMBL24258941 0.82 NR1H4 (0.50) RAB9ALMNAALDH1A1NR1H4
SCHEMBL22354184 0.81 NR1H4 (0.51) NR1H4
SCHEMBL22354110 0.76 MAPT (0.36) RAB9ALMNAALDH1A1HTTNPC1
SCHEMBL24258958 0.76 NR1H4 (0.45) NR1H4TNKSPARP1PARP2MAPT
SCHEMBL24259266 0.76 LMNA (0.43) RAB9ALMNAALDH1A1HTTKMT2A
SCHEMBL24259347 0.75 MAPT (0.37) RAB9ALMNAALDH1A1HTTNPC1
SCHEMBL24258902 0.74 NR1H4 (0.45) NR1H4
SCHEMBL24602597 0.73 ALDH1A1 (0.42) RAB9ALMNAALDH1A1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020168143-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-08-20 WO disclosed