SCHEMBL22355703

SCHEMBL22355703

Cc1ccc2c(c1)CC1(CCN(c3ccc(/C(C=N)=C/N)cc3)C1=O)N2

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.44
ITGB3 P05106 3/20 0.30
ITGA2B P08514 3/20 0.30
GAA P10253 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22355676 0.90 ROCK2 (0.43) ROCK2
SCHEMBL22355668 0.89 ROCK2 (0.42) ROCK2GAA
SCHEMBL22355688 0.85 ROCK2 (0.42) ROCK2ITGB3ITGA2B
SCHEMBL22355704 0.79 ROCK2 (0.36) ROCK2
SCHEMBL22355710 0.78 ROCK2 (0.34) ROCK2
SCHEMBL22355678 0.78 ROCK2 (0.37) ROCK2
SCHEMBL22355725 0.78 ROCK2 (0.40) ROCK2ITGB3ITGA2B
SCHEMBL22355685 0.75 ROCK2 (0.50) ROCK2
SCHEMBL22355724 0.74 ROCK2 (0.47) ROCK2
SCHEMBL22355757 0.72 ITGB3 (0.41) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481817-B1 SPIROLACTAMS AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2020-08-19 EP disclosed