SCHEMBL22355756

SCHEMBL22355756

COc1ccc2c(c1)N(C(=O)OC(C)(C)C)C(C=O)C2

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KYAT1 Q16773 1/20 0.43
KYAT3 Q6YP21 1/20 0.43
AADAT Q8N5Z0 1/20 0.43
ALDH1A1 P00352 2/20 0.40
STS P08842 2/20 0.40
EPHX2 P34913 1/20 0.39
FFAR4 Q5NUL3 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
GHSR Q92847 2/20 0.37
HTT P42858 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NR1H2 P55055 2/20 0.36
GPR119 Q8TDV5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29442994 0.82 KYAT1 (0.45) KYAT1KYAT3AADATALDH1A1STS
SCHEMBL4999428 0.82 KYAT1 (0.45) KYAT1KYAT3AADATALDH1A1STS
SCHEMBL29442988 0.81 PTPN1 (0.47) KYAT1KYAT3AADATALDH1A1STS
SCHEMBL21490330 0.81 PTPN1 (0.47) KYAT1KYAT3AADATALDH1A1STS
SCHEMBL1760532 0.81 NOTUM (0.46) ALDH1A1
SCHEMBL30390545 0.81 NOTUM (0.46) ALDH1A1
SCHEMBL30390623 0.81 NOTUM (0.46) ALDH1A1
SCHEMBL25697688 0.81 NOTUM (0.46) ALDH1A1
SCHEMBL19329216 0.81 HDAC8 (0.53) HDAC8
SCHEMBL19329217 0.81 HDAC8 (0.53) HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481817-B1 SPIROLACTAMS AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2020-08-19 EP disclosed