SCHEMBL22360326

SCHEMBL22360326

CC1(O)Cc2ccccc2CN(C2CCN(C(=O)c3cnc(N4CC5(COC5)C4)nc3)CC2)C1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 16/20 0.61
AKR1C3 P42330 1/20 0.39
DGAT2 Q96PD7 1/20 0.38
L3MBTL3 Q96JM7 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22360325 0.90 ADRA1A (0.57) ADRA1ADGAT2L3MBTL3L3MBTL1
SCHEMBL16824482 0.87 ADRA1A (0.80) ADRA1AAKR1C3
SCHEMBL16855450 0.77 ADRA1A (0.61) ADRA1A
SCHEMBL22360365 0.77 ADRA1A (0.55) ADRA1AAKR1C3DGAT2
SCHEMBL16846240 0.76 ADRA1A (1.00) ADRA1A
SCHEMBL16855449 0.76 ADRA1A (0.64) ADRA1A
SCHEMBL16827304 0.75 ADRA1A (1.00) ADRA1A
SCHEMBL22345182 0.74 ADRA1A (0.64) ADRA1ADGAT2
SCHEMBL16855262 0.74 ADRA1A (0.81) ADRA1A
SCHEMBL20052796 0.73 ADRA1A (0.79) ADRA1AL3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020165031-A1 SUBSTITUTED ISOQUINOLINE-PIPERIDINYLMETHANONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-20 WO disclosed