SCHEMBL22360365

SCHEMBL22360365

O=C(c1cnc(N2CC3(COC3)C2)nc1)N1CCC(N2C=Cc3ccccc3C2)CC1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 13/20 0.55
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
AKR1C3 P42330 1/20 0.36
DGAT2 Q96PD7 2/20 0.36
MGLL Q99685 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22360323 0.87 ADRA1A (0.41) ADRA1ADGAT2
SCHEMBL22360349 0.87 ADRA1A (0.52) ADRA1AALDH1A1HPGDHSD17B10DGAT2
SCHEMBL16824482 0.81 ADRA1A (0.80) ADRA1AAKR1C3PRMT5WDR77
SCHEMBL22360326 0.77 ADRA1A (0.61) ADRA1AAKR1C3DGAT2
SCHEMBL22345182 0.75 ADRA1A (0.64) ADRA1AALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL16855449 0.72 ADRA1A (0.64) ADRA1AALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL22345187 0.72 ADRA1A (0.53) ADRA1AALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL22345186 0.72 ADRA1A (0.55) ADRA1AALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL22360319 0.71 ADRA1A (0.51) ADRA1AALDH1A1TSHR
SCHEMBL16827304 0.71 ADRA1A (1.00) ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020165031-A1 SUBSTITUTED ISOQUINOLINE-PIPERIDINYLMETHANONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-20 WO disclosed