SCHEMBL22360345

SCHEMBL22360345

O=C(c1cnc(N2CCOCC2)nc1)N1CCC(N2Cc3ccccc3C(O)C2)CC1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 13/20 0.60
GRIN1 Q05586 1/20 0.46
GRIN2B Q13224 1/20 0.46
PIK3CA P42336 2/20 0.45
MTOR P42345 2/20 0.45
PIK3CG P48736 2/20 0.45
DGAT2 Q96PD7 1/20 0.44
L3MBTL3 Q96JM7 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ACACB O00763 1/20 0.43
ACACA Q13085 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20052796 0.86 ADRA1A (0.79) ADRA1APIK3CAMTORPIK3CGL3MBTL3
SCHEMBL22360324 0.84 ADRA1A (0.46) ADRA1AGRIN1GRIN2BDGAT2L3MBTL3
SCHEMBL22360325 0.79 ADRA1A (0.57) ADRA1APIK3CAMTORPIK3CGDGAT2
SCHEMBL20175019 0.77 ADRA1A (0.61) ADRA1A
SCHEMBL22360349 0.76 ADRA1A (0.52) ADRA1APIK3CAMTORPIK3CGDGAT2
SCHEMBL16846280 0.75 ADRA1A (1.00) ADRA1A
SCHEMBL20052743 0.75 ADRA1A (0.64) ADRA1AL3MBTL1
SCHEMBL20220382 0.74 ADRA1A (0.80) ADRA1A
SCHEMBL16855259 0.74 ADRA1A (0.80) ADRA1A
SCHEMBL16827278 0.74 ADRA1A (1.00) ADRA1ADGAT2L3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020165031-A1 SUBSTITUTED ISOQUINOLINE-PIPERIDINYLMETHANONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-20 WO disclosed