SCHEMBL22360324

SCHEMBL22360324

O=C(c1cnc(N2CC(CO)(CO)C2)nc1)N1CCC(N2Cc3ccccc3C(O)C2)CC1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 15/20 0.46
GRIN1 Q05586 1/20 0.44
GRIN2B Q13224 1/20 0.44
DGAT2 Q96PD7 1/20 0.39
L3MBTL3 Q96JM7 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22345196 0.87 ADRA1A (0.60) ADRA1A
SCHEMBL22360345 0.84 ADRA1A (0.60) ADRA1AGRIN1GRIN2BDGAT2L3MBTL3
SCHEMBL22360323 0.78 ADRA1A (0.41) ADRA1ADGAT2
SCHEMBL22360348 0.78 ADRA1A (0.57) ADRA1ADGAT2
SCHEMBL22345185 0.75 ADRA1A (0.60) ADRA1ADGAT2
SCHEMBL16824482 0.73 ADRA1A (0.80) ADRA1A
SCHEMBL20052796 0.71 ADRA1A (0.79) ADRA1AL3MBTL3L3MBTL1
SCHEMBL20220382 0.70 ADRA1A (0.80) ADRA1A
SCHEMBL16855259 0.70 ADRA1A (0.80) ADRA1A
SCHEMBL18186147 0.70 ADRA1A (0.67) ADRA1ADGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020165031-A1 SUBSTITUTED ISOQUINOLINE-PIPERIDINYLMETHANONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-20 WO disclosed