SCHEMBL22436705

SCHEMBL22436705

CCc1c(I)c(C(O)CCN2CCOCC2)nn1C

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
TSHR P16473 1/20 0.33
USP2 O75604 1/20 0.32
MCL1 Q07820 1/20 0.31
HTR7 P34969 1/20 0.30
CYP1A2 P05177 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
HTR2A P28223 1/20 0.30
MAPK1 P28482 1/20 0.30
SCN1A P35498 1/20 0.30
HTR2B P41595 1/20 0.30
KCNH2 Q12809 1/20 0.30
SCN2A Q99250 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
SCN3A Q9NY46 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22436703 1.00 ALDH1A1 (0.39) ALDH1A1KDM4ETSHRUSP2MCL1
SCHEMBL22436698 0.85 ALDH1A1 (0.39) ALDH1A1KDM4ETSHRUSP2MCL1
SCHEMBL30679099 0.85 ALDH1A1 (0.39) ALDH1A1KDM4ETSHRUSP2MCL1
SCHEMBL22436728 0.80
SCHEMBL30679120 0.79 ALDH1A1 (0.38) ALDH1A1KDM4ETSHRUSP2MCL1
SCHEMBL22436668 0.79 ALDH1A1 (0.38) ALDH1A1KDM4ETSHRUSP2MCL1
SCHEMBL22436708 0.78 KDM4E (0.34) ALDH1A1KDM4E
SCHEMBL22436707 0.78 KDM4E (0.34) ALDH1A1KDM4E
SCHEMBL22436795 0.74 ALDH1A1 (0.40) ALDH1A1KDM4ETSHRUSP2MAPK1
SCHEMBL30679119 0.74 ALDH1A1 (0.40) ALDH1A1KDM4ETSHRUSP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111757884-A Substituted macrocyclic indole derivatives 拜耳股份公司 2020-10-09 CN disclosed
EP-3710451-A1 SUBSTITUTED MACROCYCLIC INDOLE DERIVATIVES Bayer Aktiengesellschaft (DE) 2020-09-23 EP disclosed