SCHEMBL22453369

SCHEMBL22453369

CN(c1ccc(C2CCCCC2)cc1)c1cc(C2CC2)c(N)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 2/20 0.41
BACE1 P56817 1/20 0.37
ADK P55263 2/20 0.37
DGAT1 O75907 2/20 0.34
TDO2 P48775 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32
NOS2 P35228 2/20 0.32
SLC18A3 Q16572 1/20 0.32
KDM4C Q9H3R0 3/20 0.32
KDM6B O15054 1/20 0.31
CYP11B2 P19099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453569 0.86 PSMB5 (0.42) PSMB5BACE1ADKDGAT1KDM4E
SCHEMBL22452935 0.80 BACE1 (0.38) PSMB5BACE1ADKDGAT1KDM4E
SCHEMBL22453567 0.79 PSMB5 (0.45) PSMB5BACE1ADKDGAT1KDM4E
SCHEMBL22452599 0.78 PSMB5 (0.46) PSMB5BACE1ADKDGAT1KDM4E
SCHEMBL22452611 0.74 PSMB5 (0.42) PSMB5BACE1DGAT1KDM4EGLA
SCHEMBL20210323 0.72 SLC18A3 (0.46) PSMB5BACE1HTTKMT2ASMN1; SMN2
SCHEMBL22453195 0.72 SLC18A3 (0.44) PSMB5BACE1ADKKDM4EGLA
SCHEMBL22452583 0.70 S100B (0.41) PSMB5BACE1DGAT1KDM4EHTT
SCHEMBL22453700 0.69 BACE1 (0.38) PSMB5BACE1DGAT1KDM4EHTT
SCHEMBL22452582 0.67 CYP3A4 (0.43) PSMB5BACE1TDP1L3MBTL1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed