SCHEMBL22453700

SCHEMBL22453700

CN(c1ccc(C2CCCCC2)cc1)c1ccc(N)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.38
PSMB5 P28074 1/20 0.37
STAT3 P40763 2/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 1/20 0.36
APP P05067 1/20 0.36
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
SLC18A3 Q16572 1/20 0.35
MAPT P10636 3/20 0.34
LMNA P02545 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.34
HTT P42858 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 2/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22452583 0.84 S100B (0.41) BACE1PSMB5STAT3CYP3A4NOS3
SCHEMBL22452935 0.83 BACE1 (0.38) BACE1PSMB5NOS3NOS1NOS2
SCHEMBL20210323 0.81 SLC18A3 (0.46) BACE1PSMB5NOS3NOS1NOS2
SCHEMBL20800879 0.80 SLC18A3 (0.41) PSMB5STAT3CYP3A4CYP2C9APP
SCHEMBL22453195 0.80 SLC18A3 (0.44) BACE1PSMB5STAT3CYP3A4NOS3
SCHEMBL27543160 0.80 BACE1 (0.47) BACE1MAPTLMNAKMT2AALDH1A1
SCHEMBL20800878 0.78 SLC18A3 (0.42) PSMB5APPSLC18A3LMNAKMT2A
SCHEMBL30868485 0.78 ALDH1A1 (0.45) BACE1ALDH1A1HDAC1HDAC2
SCHEMBL20210026 0.76 SLC18A3 (0.41) BACE1PSMB5STAT3SLC18A3MAPT
SCHEMBL22453515 0.75 MEN1 (0.42) KMT2AGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed