SCHEMBL22453374

SCHEMBL22453374

Nc1cccc(C(=O)Nc2ccc(C3CCCCC3)cc2Cl)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66
HSD17B10 Q99714 1/20 0.66
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
MAPT P10636 1/20 0.60
SERPINE1 P05121 2/20 0.59
HDAC1 Q13547 3/20 0.52
KMO O15229 1/20 0.46
CNR1 P21554 1/20 0.44
HDAC2 Q92769 1/20 0.44
KDM4C Q9H3R0 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
DDB1 Q16531 1/20 0.42
CRBN Q96SW2 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC11 Q96DB2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14113410 0.84 SERPINE1 (0.57) MEN1KMT2AMAPTSERPINE1NPC1
SCHEMBL22453063 0.79 SERPINE1 (0.60) MEN1KMT2ASERPINE1KMONPC1
SCHEMBL22453372 0.77 GAA (0.49) SMN1; SMN2MEN1KMT2AMAPTSERPINE1
SCHEMBL22452646 0.77 SERPINE1 (0.50) SMN1; SMN2NPSR1HSD17B10MEN1KMT2A
SCHEMBL3824109 0.77 CA1 (0.48) SMN1; SMN2NPSR1HSD17B10MEN1KMT2A
SCHEMBL3769385 0.76 NPSR1 (0.80) SMN1; SMN2NPSR1HSD17B10MEN1KMT2A
SCHEMBL22453286 0.76 SERPINE1 (0.56) SMN1; SMN2MEN1KMT2AMAPTSERPINE1
SCHEMBL864819 0.76 MEN1 (1.00) SMN1; SMN2NPSR1HSD17B10MEN1KMT2A
SCHEMBL18147885 0.76 SMN1; SMN2 (0.78) SMN1; SMN2NPSR1HSD17B10MEN1KMT2A
SCHEMBL22453347 0.76 SERPINE1 (0.58) SMN1; SMN2MEN1KMT2ASERPINE1KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed