SCHEMBL22453372

SCHEMBL22453372

Nc1cccc(Nc2ccc(C3CCCCC3)cc2Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
HTT P42858 2/20 0.49
ALDH1A1 P00352 2/20 0.49
ALOX15 P16050 1/20 0.49
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GFER P55789 1/20 0.42
TDO2 P48775 1/20 0.41
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KCNH2 Q12809 2/20 0.38
CYP2D6 P10635 1/20 0.38
SERPINE1 P05121 2/20 0.38
BACE1 P56817 1/20 0.38
XBP1 P17861 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453371 0.82 ALDH1A1 (0.40) GAATDP1HTTALDH1A1ALOX15
SCHEMBL22453375 0.78 KDM1A (0.40) GAATDP1HTTALDH1A1ALOX15
SCHEMBL22453374 0.77 SMN1; SMN2 (0.66) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL22453348 0.76 KMT2A (0.42) TDP1HTTALDH1A1MEN1KMT2A
SCHEMBL22453062 0.75 DHODH (0.52) TDP1HTTALDH1A1LMNAMAPT
SCHEMBL6100303 0.75 KMO (0.53) ALDH1A1MAPTKDM4EGFERTDO2
SCHEMBL1176491 0.75 KMO (0.53) ALDH1A1MAPTKDM4EGFERTDO2
SCHEMBL21332384 0.73 KMO (0.51) GAATDP1HTTALDH1A1LMNA
SCHEMBL16334825 0.73 HDAC4 (0.52) GAATDP1ALDH1A1LMNAMAPT
SCHEMBL2652971 0.72 TDO2 (0.40) GAAHTTALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed