SCHEMBL22453375

SCHEMBL22453375

Nc1cc(Nc2ccc(C3CCCCC3)cc2Cl)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.40
CTSC P53634 1/20 0.38
DGAT1 O75907 1/20 0.37
ACLY P53396 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRB2 P47870 1/20 0.37
CNR1 P21554 2/20 0.35
CNR2 P34972 2/20 0.35
DHODH Q02127 1/20 0.35
ALDH1A1 P00352 3/20 0.35
GAA P10253 3/20 0.35
HTR2C P28335 2/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 2/20 0.35
CYP2D6 P10635 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22452932 0.84 KDM1A (0.40) KDM1AGAAHTR2CHTTMAPT
SCHEMBL22453059 0.79 AKR1C3 (0.57) KDM1AACLYCNR2DHODHALDH1A1
SCHEMBL22453372 0.78 GAA (0.49) DHODHALDH1A1GAAALOX15HTT
SCHEMBL22452643 0.77 CNR2 (0.46) KDM1ACNR2ALDH1A1MAPTCYP2D6
SCHEMBL22452817 0.77 KDM1A (0.42) KDM1ACTSCDGAT1ACLYDHODH
SCHEMBL22453371 0.74 ALDH1A1 (0.40) DHODHALDH1A1GAAALOX15HTT
SCHEMBL22452859 0.74 ALDH1A1 (0.41) CNR1CNR2ALDH1A1GAAALOX15
SCHEMBL22453849 0.71 MEN1 (0.35) CNR1CNR2ALDH1A1GAAALOX15
SCHEMBL16904557 0.68 CTSC (0.43) CTSCCNR1CNR2GAAHTT
SCHEMBL3681390 0.68 HTR2C (0.66) KDM1AHTR2CHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed