SCHEMBL22453382

SCHEMBL22453382

COc1ccc(Nc2cccc(C(=O)Nc3ccc(C4CCCCC4)cc3Cl)c2)c(C(=O)O)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 2/20 0.58
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
LMNA P02545 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
HPGD P15428 1/20 0.54
GFER P55789 1/20 0.54
AKR1C3 P42330 4/20 0.49
AKR1C2 P52895 4/20 0.49
MAPT P10636 2/20 0.48
POLB P06746 1/20 0.48
ALB P02768 1/20 0.47
NR1H4 Q96RI1 1/20 0.46
FABP3 P05413 1/20 0.46
FABP4 P15090 1/20 0.46
DHODH Q02127 2/20 0.45
CA2 P00918 1/20 0.45
ALDH1A1 P00352 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22452796 0.93 SERPINE1 (0.48) SERPINE1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL22453347 0.91 SERPINE1 (0.58) SERPINE1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL22453063 0.88 SERPINE1 (0.60) SERPINE1MEN1KMT2APOLBDHODH
SCHEMBL22452642 0.86 SERPINE1 (0.47) SERPINE1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL22452646 0.86 SERPINE1 (0.50) SERPINE1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL22453286 0.81 SERPINE1 (0.56) SERPINE1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL22452475 0.81 MEN1 (0.58) SERPINE1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL22452640 0.79 SERPINE1 (0.49) SERPINE1MEN1KMT2AMAPTALDH1A1
SCHEMBL22452719 0.77 DHODH (0.51) MEN1KMT2ALMNASMN1; SMN2HPGD
SCHEMBL22453374 0.76 SMN1; SMN2 (0.66) SERPINE1MEN1KMT2ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed