SCHEMBL2245494

SCHEMBL2245494

NC(=O)CC[C@H](NC(=O)c1ccc(-c2cccs2)cc1)C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 3/20 0.65
CA2 P00918 5/20 0.58
CA1 P00915 3/20 0.58
MMP12 P39900 1/20 0.53
CTSB P07858 1/20 0.50
CTSS P25774 1/20 0.50
C3AR1 Q16581 1/20 0.46
KMT2A Q03164 1/20 0.45
MMP2 P08253 2/20 0.44
MMP9 P14780 2/20 0.44
MRGPRX4 Q96LA9 1/20 0.43
HDAC1 Q13547 1/20 0.43
DRD2 P14416 2/20 0.43
DRD4 P21917 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2248320 0.91 HPGDS (0.54) HPGDSCA2CA1MMP12C3AR1
SCHEMBL2245488 0.86 HPGDS (0.71) HPGDSCA2CA1MMP12CTSB
SCHEMBL2246061 0.85 CA2 (0.69) HPGDSCA2CA1MMP12C3AR1
SCHEMBL2245325 0.85 CA2 (0.69) HPGDSCA2CA1MMP12C3AR1
SCHEMBL4384045 0.81 CA2 (0.53) CA2CA1CTSBCTSSKMT2A
SCHEMBL2248627 0.81 CA2 (0.60) CA2CA1MMP12C3AR1KMT2A
SCHEMBL5260684 0.80 CA2 (0.70) CA2CA1C3AR1KMT2AMMP2
SCHEMBL5260686 0.80 CA2 (0.70) CA2CA1C3AR1KMT2AMMP2
SCHEMBL2249747 0.80 CA2 (0.63) CA2CA1MMP12C3AR1KMT2A
SCHEMBL27708431 0.80 CA2 (0.57) HPGDSCA2CA1MMP12C3AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101223130-A Glutamate aggrecanase inhibitors WYETH CORP (US) 2008-07-16 CN claimed
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed
CN-101223130-A Glutamate aggrecanase inhibitors WYETH CORP (US) 2008-07-16 CN disclosed