SCHEMBL22462090

SCHEMBL22462090

CS(=O)(=O)N1CCC(N2C[C](n3cc(-c4ncnc5[nH]ccc45)cn3)C2)CC1

nearest known ligand 0.65

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 16/20 0.65
JAK1 P23458 11/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22462089 0.92 JAK1 (0.66) JAK2JAK1
SCHEMBL22462086 0.90 JAK2 (0.66) JAK2JAK1
SCHEMBL14563734 0.87 JAK2 (0.52) JAK2JAK1
SCHEMBL27182358 0.86 JAK2 (0.51) JAK2JAK1
SCHEMBL14563805 0.85 JAK2 (0.65) JAK2JAK1
SCHEMBL14563845 0.85 JAK2 (0.50) JAK2JAK1
SCHEMBL28466379 0.85 JAK2 (0.66) JAK2JAK1
SCHEMBL14563676 0.85 JAK2 (0.69) JAK2JAK1
SCHEMBL14563857 0.84 JAK2 (0.53) JAK2JAK1
SCHEMBL17387434 0.81 JAK2 (0.65) JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3715347-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS Incyte Holdings Corporation (US) 2020-09-30 EP claimed
EP-3715347-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS Incyte Holdings Corporation (US) 2020-09-30 EP disclosed