SCHEMBL22471072

SCHEMBL22471072

COc1cc(N2CCC(N3CCOCC3)CC2)c([N+](=O)[O-])cc1Br

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 12/20 0.48
ALDH1A1 P00352 7/20 0.48
HTT P42858 2/20 0.48
LMNA P02545 2/20 0.48
GAA P10253 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
S1PR1 P21453 1/20 0.47
POLB P06746 2/20 0.43
TP53 P04637 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
MAPK1 P28482 3/20 0.42
TDP1 Q9NUW8 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29757727 0.91 MAPT (0.46) MAPTALDH1A1HTTLMNAGAA
SCHEMBL23421504 0.91 MAPT (0.46) MAPTALDH1A1HTTLMNAGAA
SCHEMBL22470985 0.90 KDM4E (0.46) MAPTALDH1A1LMNAS1PR1POLB
SCHEMBL22471057 0.89 KDM4E (0.46) MAPTALDH1A1HTTLMNANPSR1
SCHEMBL22471048 0.89 HTT (0.54) MAPTALDH1A1HTTLMNAGAA
SCHEMBL22471036 0.89 HTT (0.54) MAPTALDH1A1HTTLMNAGAA
SCHEMBL22471075 0.88 SIRT6 (0.46) MAPTALDH1A1LMNAPOLBTP53
SCHEMBL22595700 0.88 MAPT (0.43) MAPTALDH1A1HTTLMNAGAA
SCHEMBL22471254 0.87 MAPT (0.42) MAPTALDH1A1LMNAGAAS1PR1
SCHEMBL28673273 0.87 MAPT (0.48) MAPTALDH1A1HTTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111356687-B Pyrimidine-containing tri-substituted imidazole compound and application thereof 广州必贝特医药技术有限公司 2021-03-30 CN disclosed
WO-2020192302-A1 PYRIMIDINE-CONTAINING TRI-SUBSTITUTED IMIDAZOLE COMPOUND AND APPLICATION THEREOF 广州必贝特医药技术有限公司 2020-10-01 WO disclosed
CN-111356687-A Pyrimidine-containing tri-substituted imidazole compound and application thereof 广州必贝特医药技术有限公司 2020-06-30 CN disclosed