SCHEMBL2248046

SCHEMBL2248046

[c]1c(-c2nccc3ccccc23)ncc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.42
MAPT P10636 5/20 0.42
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
KMT2A Q03164 2/20 0.42
GLA P06280 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PLAU P00749 2/20 0.41
CYP2A6 P11509 1/20 0.41
F12 P00748 1/20 0.41
NCF1 P14598 1/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
BACE1 P56817 1/20 0.41
GPR55 Q9Y2T6 1/20 0.39
MAPK1 P28482 3/20 0.37
CYP3A4 P08684 3/20 0.37
LMNA P02545 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL467327 0.75 MAPT (0.43) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL199273 0.74 PLAU (0.60) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL29923403 0.74 PLAU (0.60) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL30522769 0.72 PLAU (0.58) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL12223316 0.70 PLAU (0.56) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL13978866 0.70 PLAU (0.56) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL158912 0.70 BCHE (0.58) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL29986041 0.70 BCHE (0.58) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL12112873 0.69 MAPT (0.58) KDM4EMAPTNPC1RAB9AL3MBTL1
SCHEMBL21810846 0.69 MAPT (0.43) KDM4EMAPTNPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105308026-A Cyclic azine compound having adamantyl group, production method, and organic electroluminescent element containing said compound as constituent TOSOH CORP 2016-02-03 CN disclosed
EP-2341775-A1 INHIBITORS OF JANUS KINASES Merck & Co., Inc. (US) 2011-07-13 EP disclosed
WO-2010014453-A1 INHIBITORS OF JANUS KINASES MERCK & CO., INC. (US) 2010-02-04 WO disclosed
EP-1037868-B1 $g(a)-HYDROXY, -AMINO, AND HALO DERIVATIVES OF $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS UPJOHN CO (US) 2003-02-05 EP disclosed