SCHEMBL22481385

SCHEMBL22481385

CC(C)(C)OC(=O)N[C@H]1CCCN(c2nc3ccccc3[nH]2)C1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.54
MAP4K4 O95819 2/20 0.53
BTK Q06187 3/20 0.49
JAK3 P52333 1/20 0.49
AURKA O14965 3/20 0.49
PDPK1 O15530 3/20 0.49
AURKB Q96GD4 3/20 0.49
BCHE P06276 2/20 0.47
PARP1 P09874 2/20 0.47
ACHE P22303 1/20 0.47
TRPC3 Q13507 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
OPRK1 P41145 1/20 0.46
OGFRL1 Q5TC84 1/20 0.46
KIF18A Q8NI77 1/20 0.45
PIM1 P11309 1/20 0.44
PIM3 Q86V86 1/20 0.44
PIM2 Q9P1W9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22481485 1.00 PDE10A (0.54) PDE10AMAP4K4BTKJAK3AURKA
SCHEMBL29668378 1.00 PDE10A (0.54) PDE10AMAP4K4BTKJAK3AURKA
SCHEMBL29668374 1.00 PDE10A (0.54) PDE10AMAP4K4BTKJAK3AURKA
SCHEMBL22464692 0.84 BCHE (0.54) BCHEACHETRPC3
SCHEMBL22481577 0.83 TRPC3 (0.48) BCHETRPC3OPRM1OPRD1OPRK1
SCHEMBL29668327 0.83 TRPC3 (0.48) BCHETRPC3OPRM1OPRD1OPRK1
SCHEMBL29668159 0.83 TRPC3 (0.48) BCHETRPC3OPRM1OPRD1OPRK1
SCHEMBL22481378 0.83 TRPC3 (0.48) BCHETRPC3OPRM1OPRD1OPRK1
SCHEMBL22481501 0.80 BCHE (0.45) BCHEACHETRPC3
SCHEMBL29668300 0.80 BCHE (0.45) BCHEACHETRPC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11332459-B2 Benzimidazole derivatives and their uses TEIJIN PHARMA LIMITED (JP) 2022-05-17 US disclosed
US-20200308145-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USES AMGEN INC. (US) 2020-10-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200308145-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USES TRPC6, TRPV6, TRPM6 PDE10A 1273/4885MAP4K4 1473/4885BTK 290/4885
US-11332459-B2 Benzimidazole derivatives and their uses TRPC6, TRPV6, TRPM6 PDE10A 1273/4885MAP4K4 1473/4885BTK 290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.