SCHEMBL22491591

SCHEMBL22491591

CC(C)(C)OC(=O)N1CCC(c2c[nH]c3cc(C4(Cl)CC4)ccc23)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
BRD4 O60885 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
CREBBP Q92793 1/20 0.45
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
HSD11B1 P28845 3/20 0.42
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
JAK3 P52333 1/20 0.42
SCN9A Q15858 1/20 0.41
CNR1 P21554 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PTPN2 P17706 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN6 P29350 1/20 0.40
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771971 0.85 AVPR1A (0.50) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL12127425 0.85 KDM4E (0.49) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL4882143 0.83 DRD2 (0.56) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL557776 0.80 KDM4E (0.70) KDM4EBRD4ALDH1A1POLBCREBBP
Hydrochloric Acid SCHEMBL1703924 0.79 KDM4E (0.68) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL892836 0.79 OPRM1 (0.53) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL30567991 0.79 OPRM1 (0.53) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL12127418 0.79 KDM4E (0.49) KDM4EBRD4ALDH1A1POLBCREBBP
Hydrochloric Acid SCHEMBL1703941 0.78 OPRM1 (0.52) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL8618496 0.77 CYP1A2 (0.63) KDM4EBRD4ALDH1A1POLBCREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3717477-A1 NEW HETEROCYCLIC COMPOUNDS H. Hoffnabb-La Roche Ag (CH) 2020-10-07 EP disclosed