Benzoquinone

Benzoquinone

SCHEMBL22491815

C[C@H]([C@H](C(=O)O)c1ccc(Cl)cc1)C(F)(F)F.O=C1C=CC(=O)C=C1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 10/20 0.42
PRCP P42785 2/20 0.38
POLB P06746 1/20 0.38
PPARG P37231 3/20 0.36
BRD4 O60885 1/20 0.36
GRN P28799 1/20 0.35
SORT1 Q99523 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1906571 0.92 FFAR2 (0.47) FFAR2PRCPPOLBPPARGBRD4
SCHEMBL1905489 0.92 FFAR2 (0.47) FFAR2PRCPPOLBPPARGBRD4
SCHEMBL9899646 0.92 FFAR2 (0.47) FFAR2PRCPPOLBPPARGBRD4
SCHEMBL22491784 0.92 FFAR2 (0.47) FFAR2PRCPPOLBPPARGBRD4
SCHEMBL14798252 0.82 CYP2D6 (0.46) FFAR2POLB
SCHEMBL1932498 0.82 CYP2D6 (0.46) FFAR2POLB
SCHEMBL1905993 0.80 FFAR2 (0.47) FFAR2PRCPBRD4
SCHEMBL1907199 0.80 FFAR2 (0.47) FFAR2PRCPBRD4
SCHEMBL24893827 0.79 AKR1C3 (0.46) PPARGGRNSORT1
SCHEMBL24893812 0.79 AKR1C3 (0.46) PPARGGRNSORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3717480-A1 METHOD FOR PRODUCING (3S)-3-(4-CHLOR-3-{[(2S,3R)-2-(4-CHLORPHENYL)-4,4,4-TRIFLUOR-3-METHYLBUTANOYL]AMINO}PHENYL)-3-CYCLO-PROPYLPROPANOIC ACID AND THE CRYSTALLINE FORM THEREOF FOR USE AS A PHARMACEUTICAL INGREDIENT Bayer Pharma Aktiengesellschaft (DE) 2020-10-07 EP disclosed
CN-111433204-A Process for the preparation of (3S) -3- (4-chloro-3- { [ (2S,3R) -2- (4-chlorophenyl) -4,4, 4-trifluoro-3-methylbutyryl ] amino } phenyl) -3-cyclopropylpropionic acid and crystalline forms thereof for use as a pharmaceutically active substance 拜耳制药股份公司 2020-07-17 CN disclosed