SCHEMBL22492296

SCHEMBL22492296

NS(=O)(=O)C1NCc2ccccc2N1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMYD3 Q9H7B4 1/20 0.34
PRCP P42785 1/20 0.33
PNMT P11086 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3139036 0.75 GAA (0.47) GAAMAPTCA1CA2SMYD3
SCHEMBL2658519 0.74 GAA (0.46) GAAMAPTMEN1KMT2ASMYD3
SCHEMBL517885 0.72 SMYD3 (0.43) GAAMAPTCA1CA2SMYD3
SCHEMBL31634875 0.72 SMYD3 (0.43) GAAMAPTCA1CA2SMYD3
SCHEMBL3468367 0.72 MEN1 (0.40) GAAMAPTMEN1KMT2APRCP
SCHEMBL31145667 0.72 MEN1 (0.40) GAAMAPTMEN1KMT2APRCP
SCHEMBL26606581 0.71
Carbamic Acid SCHEMBL1271067 0.70 SMYD3 (0.44) GAAMAPTCA1CA2KMT2A
SCHEMBL19676469 0.70 PNMT (0.41) GAAMAPTMEN1KMT2APRCP
SCHEMBL27678136 0.69 PNMT (0.50) CA1CA2PRCPPNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154913-A1 INHIBITORS OF PARG ARASE THERAPEUTICS INC. (US) 2023-08-17 WO claimed
CN-105272904-B N- phenylamide compound and its application 中国科学院广州生物医药与健康研究院 2019-04-09 CN claimed
WO-2024023330-A1 SUBSTITUTED BICYCLIC HETEROARYL SULFONAMIDE DERIVATIVES FOR THE TREATMENT OF CANCER NODUS ONCOLOGY LIMITED (GB) 2024-02-01 WO disclosed
WO-2023175185-A1 2,4-DIOXO-1,4-DIHYDROQUINAZOLINE DERIVATIVES AS PARG INHIBITORS FOR THE TREATMENT OF CANCER FORX THERAPEUTICS AG (CH) 2023-09-21 WO disclosed
WO-2023175184-A1 2,4-DIOXO-1,4-DIHYDROQUINAZOLINE DERIVATIVES AS PARG INHIBITORS FOR THE TREATMENT OF CANCER FORX THERAPEUTICS AG (CH) 2023-09-21 WO disclosed
WO-2023154913-A1 INHIBITORS OF PARG ARASE THERAPEUTICS INC. (US) 2023-08-17 WO disclosed
EP-3716968-A1 SIGMA-1 RECEPTOR AGONIST SYSTOLIC BLOOD PRESSURE THERAPY Anavex Life Sciences Corp. (US) 2020-10-07 EP disclosed