SCHEMBL3468367

SCHEMBL3468367

NC1NCc2ccccc2N1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
PRCP P42785 1/20 0.37
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PNMT P11086 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31145667 1.00 MEN1 (0.40) MEN1KMT2AGAAMAPTPRCP
SCHEMBL19676469 0.77 PNMT (0.41) MEN1KMT2AGAAMAPTPRCP
SCHEMBL6075506 0.75 GAA (0.43) MEN1KMT2AGAAMAPTPRCP
SCHEMBL29239505 0.75 MEN1 (0.40) MEN1KMT2AGAAMAPTPRCP
SCHEMBL1436282 0.75 MEN1 (0.40) MEN1KMT2AGAAMAPTPRCP
SCHEMBL14730122 0.75 ALOX15 (0.41) MEN1KMT2AGAAMAPTPRCP
SCHEMBL9672402 0.75 MEN1 (0.41) MEN1KMT2AGAAMAPTALOX15
SCHEMBL17454501 0.73 CHRNB2 (0.35)
SCHEMBL2658519 0.73 GAA (0.46) MEN1KMT2AGAAMAPTPRCP
SCHEMBL9955369 0.73 CHRNB2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108018037-B 6, 8-methano tetrahydroquinazoline-2-amine Schiff base type iron ion fluorescent probe and preparation method and application thereof 南京林业大学 2020-01-24 CN claimed
CN-108018037-A 6,8- endo-methylene group tetrahydro quinazoline -2- amine Schiff bases iron ion fluorescence probes and its preparation method and application 南京林业大学 2018-05-11 CN claimed
CN-105085413-B Tetrahydroquinazoline-2-schiff base compounds as well as synthesis method and application thereof 南京林业大学 2017-05-10 CN claimed
CN-105085413-A Tetrahydroquinazoline-2-schiff base compounds as well as synthesis method and application thereof UNIV NANJING FORESTRY 2015-11-25 CN claimed
CN-116165186-A In-situ fluorescence chromogenic reaction dual-mode detection Cu based on dopamine and isophthaol 2+ And Ag + Is a method of (2) 南昌航空大学 2023-05-26 CN disclosed
CN-108018037-A 6,8- endo-methylene group tetrahydro quinazoline -2- amine Schiff bases iron ion fluorescence probes and its preparation method and application 南京林业大学 2018-05-11 CN disclosed
CN-108018037-A 6,8- endo-methylene group tetrahydro quinazoline -2- amine Schiff bases iron ion fluorescence probes and its preparation method and application 南京林业大学 2018-05-11 CN disclosed
CN-105085413-B Tetrahydroquinazoline-2-schiff base compounds as well as synthesis method and application thereof 南京林业大学 2017-05-10 CN disclosed
CN-105085413-A Tetrahydroquinazoline-2-schiff base compounds as well as synthesis method and application thereof UNIV NANJING FORESTRY 2015-11-25 CN disclosed
WO-2012085166-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO disclosed
US-20100298289-A1 HETEROBICYCLIC COMPOUNDS AS HISTAMINE H4-RECEPTOR ANTAGONISTS UCB PHARMA, S.A. (BE) 2010-11-25 US disclosed
WO-2010072829-A1 SELECTIVE HISTAMINE H4 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF VESTIBULAR DISORDERS. INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2010-07-01 WO disclosed
US-20050197350-A1 Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof TAISHO PHARMACEUTICAL CO., LTD. 2005-09-08 US disclosed
WO-2004087669-A1 NOVEL QUINOLINE, TETRAHYDROQUINAZOLINE, AND PYRIMIDINE DERIVATIVES AND METHODS OF TREATMENT RELATED TO THE USE THEREOF TAISHO PHARMACEUTICAL CO. LTD. (JP) 2004-10-14 WO disclosed
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197350-A1 Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof HCRTR2, MCHR1, MCHR2 MEN1 734/4885KMT2A 693/4885GAA 484/4885
US-20100298289-A1 HETEROBICYCLIC COMPOUNDS AS HISTAMINE H4-RECEPTOR ANTAGONISTS HRH4, HRH2, HRH3 MEN1 1111/4885KMT2A 802/4885GAA 3320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.