SCHEMBL22497428

SCHEMBL22497428

COC(=O)c1ccccc1NC(=O)CCc1ccccc1C(F)(F)F

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.63
GAA P10253 2/20 0.59
KMT2A Q03164 2/20 0.58
POLB P06746 2/20 0.57
ALDH1A1 P00352 5/20 0.54
HTT P42858 1/20 0.54
MAPK10 P53779 2/20 0.52
MAPK8 P45983 1/20 0.52
MAPK9 P45984 1/20 0.52
HSD17B10 Q99714 3/20 0.51
TSHR P16473 1/20 0.50
MAPT P10636 1/20 0.49
LMNA P02545 1/20 0.49
RBP4 P02753 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
MEN1 O00255 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27546648 0.86 GAA (0.65) GAAKMT2APOLBALDH1A1LMNA
SCHEMBL8691586 0.82 ALDH1A1 (0.70) KDM4EGAAKMT2APOLBALDH1A1
SCHEMBL22497429 0.81 KDM4E (0.74) KDM4EGAAKMT2APOLBALDH1A1
SCHEMBL16127720 0.80 GAA (0.62) KDM4EGAAKMT2APOLBALDH1A1
SCHEMBL7108471 0.78 KDM4E (1.00) KDM4EGAAKMT2APOLBALDH1A1
SCHEMBL4797746 0.77 KMT2A (0.73) KDM4EGAAKMT2APOLBALDH1A1
SCHEMBL21015416 0.76 EPHX2 (0.51) KDM4EGAAPOLBALDH1A1HTT
SCHEMBL28057817 0.76 GAA (0.52) GAAKMT2APOLBALDH1A1MEN1
SCHEMBL27519885 0.75 GRIK1 (0.55) KDM4EGAAKMT2APOLBHSD17B10
SCHEMBL28373311 0.75 KDM4E (0.59) KDM4EKMT2APOLBALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111763164-A Preparation method and application of ortho-carbonyl amino substituted benzene derivatives 中国医学科学院药物研究所 2020-10-13 CN disclosed
WO-2020199945-A1 ORTHO-CARBONYL AMINO-SUBSTITUTED BENZENE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 中国医学科学院药物研究所 2020-10-08 WO disclosed