SCHEMBL22498482

SCHEMBL22498482

COc1ccc(NC(=N)c2ccccc2OCc2ccccc2)cc1Br

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.52
GAA P10253 3/20 0.49
CTSV O60911 2/20 0.49
CTSL P07711 2/20 0.49
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPT P10636 3/20 0.47
KDM4E B2RXH2 2/20 0.47
THRB P10828 1/20 0.47
BLM P54132 1/20 0.47
LMNA P02545 3/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
ALOX12 P18054 1/20 0.47
SGMS2 Q8NHU3 1/20 0.46
F2 P00734 1/20 0.46
F10 P00742 1/20 0.46
PRSS1 P07477 1/20 0.46
F7 P08709 1/20 0.46
MRGPRX1 Q96LB2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22498535 0.91 LRRK2 (0.49) LRRK2GAACTSVCTSLMEN1
SCHEMBL22498433 0.89 LRRK2 (0.48) LRRK2GAACTSVCTSLMEN1
SCHEMBL22498469 0.87 LRRK2 (0.46) LRRK2GAACTSVCTSLMEN1
SCHEMBL22498654 0.85 NPC1 (0.51) LRRK2GAAMEN1KMT2AMAPT
SCHEMBL22498458 0.83 NPC1 (0.51) LRRK2GAAMEN1KMT2AMAPT
SCHEMBL22498588 0.82 LRRK2 (0.54) LRRK2GAAMEN1KMT2AALDH1A1
SCHEMBL22498585 0.82 LRRK2 (0.54) LRRK2CTSVCTSLMEN1KMT2A
SCHEMBL22498480 0.82 GAA (0.60) LRRK2GAAMEN1KMT2AALDH1A1
SCHEMBL22498539 0.80 MAPT (0.48) LRRK2GAAMEN1KMT2AMAPT
SCHEMBL22498776 0.79 LRRK2 (0.59) LRRK2GAACTSVCTSLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020201305-A1 4-(2,4-BIS(2-HYDROXYPHENYL)-1H-IMIDAZOL-1-YL)BENZOIC ACID DERIVATIVES AS NOVEL IRON CHELATORS VIFOR (INTERNATIONAL) AG (CH) 2020-10-08 WO disclosed
WO-2020201305-A1 4-(2,4-BIS(2-HYDROXYPHENYL)-1H-IMIDAZOL-1-YL)BENZOIC ACID DERIVATIVES AS NOVEL IRON CHELATORS VIFOR (INTERNATIONAL) AG (CH) 2020-10-08 WO disclosed