SCHEMBL22498535

SCHEMBL22498535

COc1cc(NC(=N)c2ccccc2OCc2ccccc2)ccc1Br

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.49
CTSV O60911 3/20 0.49
CTSL P07711 3/20 0.49
GAA P10253 2/20 0.49
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
THRB P10828 1/20 0.47
BLM P54132 1/20 0.47
LMNA P02545 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
ALOX12 P18054 1/20 0.47
GRM4 Q14833 1/20 0.46
SGMS2 Q8NHU3 1/20 0.46
HTT P42858 1/20 0.46
HSD17B10 Q99714 1/20 0.46
C5AR1 P21730 1/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22498482 0.91 LRRK2 (0.52) LRRK2CTSVCTSLGAAMEN1
SCHEMBL22498458 0.85 NPC1 (0.51) LRRK2GAAMEN1KMT2AMAPT
SCHEMBL22498654 0.83 NPC1 (0.51) LRRK2GAAMEN1KMT2AMAPT
SCHEMBL22498433 0.83 LRRK2 (0.48) LRRK2CTSVCTSLGAAMEN1
SCHEMBL22498539 0.82 MAPT (0.48) LRRK2GAAMEN1KMT2AMAPT
SCHEMBL22498588 0.82 LRRK2 (0.54) LRRK2GAAMEN1KMT2AMAPT
SCHEMBL22498480 0.82 GAA (0.60) LRRK2GAAMEN1KMT2AMAPT
SCHEMBL22498469 0.80 LRRK2 (0.46) LRRK2CTSVCTSLGAAMEN1
SCHEMBL22498585 0.80 LRRK2 (0.54) LRRK2CTSVCTSLMEN1KMT2A
SCHEMBL22498776 0.76 LRRK2 (0.59) LRRK2CTSVCTSLGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020201305-A1 4-(2,4-BIS(2-HYDROXYPHENYL)-1H-IMIDAZOL-1-YL)BENZOIC ACID DERIVATIVES AS NOVEL IRON CHELATORS VIFOR (INTERNATIONAL) AG (CH) 2020-10-08 WO disclosed
WO-2020201305-A1 4-(2,4-BIS(2-HYDROXYPHENYL)-1H-IMIDAZOL-1-YL)BENZOIC ACID DERIVATIVES AS NOVEL IRON CHELATORS VIFOR (INTERNATIONAL) AG (CH) 2020-10-08 WO disclosed