SCHEMBL22508496

SCHEMBL22508496

CC(C)[C@H]1c2ccc(F)cc2CSc2cc(F)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.38
CHEK2 O96017 1/20 0.38
CDK1 P06493 1/20 0.38
PIM1 P11309 1/20 0.38
FGFR1 P11362 1/20 0.38
CDK2 P24941 1/20 0.38
MARK3 P27448 1/20 0.38
CSNK2A1 P68400 1/20 0.38
MARK2 Q7KZI7 1/20 0.38
HSD17B3 P37058 1/20 0.36
SRD5A1 P18405 3/20 0.33
NOTUM Q6P988 1/20 0.33
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22508495 1.00 AURKA (0.38) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL10444190 0.90 HSD17B3 (0.42) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL22508372 0.90 ALDH1A1 (0.38) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL10443992 0.90 ALDH1A1 (0.38) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL20101895 0.90 ALDH1A1 (0.38) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL10444152 0.79 AURKA (0.40) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL10444032 0.79 SRD5A1 (0.44) SRD5A1NOTUMSLC6A2SLC6A4SLC6A3
SCHEMBL10444154 0.78 ALDH1A1 (0.41) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL10444069 0.78 ALDH1A1 (0.41) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL10444531 0.78 SLC6A2 (0.30) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020205832-A1 FUSED POLYCYCLIC PYRIDONE COMPOUNDS AS INFLUENZA VIRUS REPLICATION INHIBITORS NIKANG THERAPEUTICS, INC. (US) 2020-10-08 WO disclosed
WO-2020205835-A1 FUSED POLYCYCLIC PYRIDONE COMPOUNDS AS INFLUENZA VIRUS REPLICATION INHIBITORS NIKANG THERAPEUTICS, INC. (US) 2020-10-08 WO disclosed