Nabumetone

Nabumetone

SCHEMBL2256

COc1ccc2cc(CCC(C)=O)ccc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGS2

The experimentally established mechanism targets of Nabumetone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 known ✓ P35354 1/20 0.58
CYP1A2 P05177 2/20 1.00
KDM4E B2RXH2 2/20 1.00
LMNA P02545 2/20 1.00
MAPT P10636 2/20 1.00
NPC1 O15118 1/20 1.00
TP53 P04637 1/20 1.00
CYP3A4 P08684 1/20 1.00
MAOA P21397 1/20 1.00
SLC6A2 P23975 1/20 1.00
RAB9A P51151 1/20 1.00
SLC6A3 Q01959 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
PTGS1 P23219 1/20 0.61
AKR1C3 P42330 1/20 0.61
AKR1C2 P52895 1/20 0.61
HCAR2 Q8TDS4 1/20 0.55
F2RL1 P55085 1/20 0.51
HSD17B1 P14061 1/20 0.50
HSD17B2 P37059 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nabumetone SCHEMBL29373228 1.00 CYP1A2 (1.00) CYP1A2KDM4ELMNAMAPTNPC1
Nabumetone SCHEMBL29570823 1.00 CYP1A2 (1.00) CYP1A2KDM4ELMNAMAPTNPC1
Nabumetone SCHEMBL3853067 1.00 CYP1A2 (1.00) CYP1A2KDM4ELMNAMAPTNPC1
Nabumetone SCHEMBL28775077 0.98 CYP1A2 (0.97) CYP1A2KDM4ELMNAMAPTNPC1
Nabumetone SCHEMBL104942 0.98 CYP1A2 (0.97) CYP1A2KDM4ELMNAMAPTNPC1
Nabumetone SCHEMBL23064140 0.97 CYP1A2 (0.94) CYP1A2KDM4ELMNAMAPTNPC1
Nabumetone SCHEMBL7554060 0.95 CYP1A2 (0.91) CYP1A2KDM4ELMNAMAPTNPC1
Nabumetone SCHEMBL3362072 0.93 RAB9A (0.86) CYP1A2KDM4ELMNAMAPTNPC1
Nabumetone SCHEMBL2325715 0.91 CYP1A2 (0.83) CYP1A2KDM4ELMNAMAPTNPC1
SCHEMBL17288829 0.90 CYP1A2 (0.82) CYP1A2KDM4ELMNAMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 58523 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747263-A1 LIPID NANOPARTICLES AND USES THEREOF University of Connecticut (US) 2026-05-27 EP claimed
US-20260139030-A1 CHIMERIC PROTEINS FOR TREATING CUTANEOUS INFLAMMATION SHATTUCK LABS INC (US) 2026-05-21 US claimed
US-20260137680-A1 NOVEL COMPOUNDS SITRYX THERAPEUTICS LTD (GB) 2026-05-21 US claimed
US-20260138973-A1 SUBSTITUTED PYRIDINES FOR USE IN TREATING OR PREVENTING INFLAMMATORY DISEASES OR DISEASES ASSOCIATED WITH AN UNDESIRABLE IMMUNE RESPONSE SITRYX THERAPEUTICS LTD (GB) 2026-05-21 US claimed
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
US-20260130928-A1 COMBINATION OF AKR1C3 ACTIVATED ANTICANCER PRODRUG COMPOUND AND ANALGESIC DRUG FOR TREATING CANCER PATIENTS ACCOMPANIED BY PAIN ASCENTAWITS PHARMACEUTICALS LTD (CN) 2026-05-14 US claimed
CN-122028914-A Combination therapy for autoimmune disorders 拜奥海芬治疗学有限公司 2026-05-12 CN claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260115209-A1 COMBINATION THERAPY INCLUDING COX-2 INHIBITOR FOR THE TREATMENT OF CANCER UNIV CALIFORNIA (US) 2026-04-30 US claimed
US-12605432-B2 Combinations for antigen based therapy DIAMYD MEDICAL AB (SE) 2026-04-21 US claimed
US-4420639-A Aromatic compounds BEECHAM GROUP LIMITED (GB) 1983-12-13 US claimed
EP-0043136-B1 CUTTING DISK PROVIDED WITH PIGMENTS HELIOTRONIC Forschungs- und Entwicklungsgesellschaft für Solarzellen-Grundstoffe mbH (DE) 1983-11-30 EP claimed
EP-0003643-B1 PROCESS FOR THE PREPARATION OF 4-(6-METHOXY-2-NAPHTHYL)-BUTAN-2-ONE; 4-(6-METHOXY-2-NAPHTHYL)-4-HYDROXYBUT-3-EN-2-ONE AND A PROCESS FOR ITS PREPARATION BEECHAM GROUP PLC (GB) 1982-09-29 EP claimed
US-4341239-A Combination check-overpressure relief valve VERNAY LABORATORIES, INC. (US) 1982-07-27 US claimed
US-4312359-A Noninvasive blood pressure measuring system LIFE CARE SYSTEMS, INC. (US) 1982-01-26 US claimed
US-4222725-A Electro-hydraulic ram control apparatus SOLID CONTROLS, INC. (US) 1980-09-16 US claimed
US-4221741-A Preparation of 4(6'-methoxy-2'-naphthyl)butan-2-one BEECHAM GROUP LIMITED (GB) 1980-09-09 US claimed
EP-0003643-A1 Process for the preparation of 4-(6-methoxy-2-naphthyl)-butan-2-one; 4-(6-methoxy-2-naphthyl)-4-hydroxybut-3-en-2-one and a process for its preparation BEECHAM GROUP PLC (GB) 1979-08-22 EP claimed
US-4075840-A Brake and steering system CLARK EQUIPMENT COMPANY (US) 1978-02-28 US claimed
US-4027482-A Variable ratio hydraulic master-cylinder ABRED ESTABLISHMENT (IT) 1977-06-07 US claimed