SCHEMBL22562215

SCHEMBL22562215

Cc1cc(C)cc(-c2ccc3c(c2)c2cc(-c4cc(C)cc(C)c4)ccc2n3-c2cc(-c3cccc(-c4ccccc4)n3)c(-n3c4ccc(-c5cc(C)cc(C)c5)cc4c4cc(-c5cc(C)cc(C)c5)ccc43)cc2C#N)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
MAPT P10636 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TGFBR1 P36897 1/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 2/20 0.37
NPSR1 Q6W5P4 2/20 0.35
HPGD P15428 1/20 0.35
PPARG P37231 1/20 0.35
NCOA2 Q15596 1/20 0.35
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP3A4 P08684 1/20 0.35
ALDH1A3 P47895 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
SQOR Q9Y6N5 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562216 0.93 KDM4E (0.41) KDM4EMAPTL3MBTL1TGFBR1ADORA2A
SCHEMBL22562217 0.92 KDM4E (0.36) KDM4EMAPTL3MBTL1TGFBR1ADORA2A
SCHEMBL22562214 0.92 KDM4E (0.38) KDM4EMAPTL3MBTL1TGFBR1ADORA2A
SCHEMBL19913243 0.91 ADORA2A (0.38) KDM4EMAPTL3MBTL1ADORA2AADORA1
SCHEMBL22562347 0.89 CYP11B1 (0.36) KDM4EMAPTL3MBTL1TGFBR1NPSR1
SCHEMBL19913244 0.89 ADORA2A (0.37) KDM4EMAPTL3MBTL1ADORA2AADORA1
SCHEMBL23487629 0.89 KDM4E (0.38) KDM4EMAPTL3MBTL1ADORA2AADORA1
SCHEMBL22562239 0.89 ALDH1A3 (0.39) KDM4EMAPTL3MBTL1TGFBR1ADORA2A
SCHEMBL22562475 0.88 KDM4E (0.41) KDM4EMAPTL3MBTL1TGFBR1ADORA2A
SCHEMBL23487627 0.87 CYP1A2 (0.37) KDM4EMAPTL3MBTL1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3418278-B1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2020-10-21 EP disclosed