SCHEMBL22600148

SCHEMBL22600148

CC(C)CCN1CCC(CC2CCN(C(C)(C)C)CC2)CC1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ARG1 P05089 1/20 0.35
ARG2 P78540 1/20 0.35
CHRM4 P08173 2/20 0.33
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
NPY1R P25929 1/20 0.30
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22600212 0.84 ACHE (0.35) ARG1ARG2CHRM4NOS3NOS1
SCHEMBL19788224 0.80 ARG1 (0.32) ARG1ARG2
SCHEMBL14102866 0.80 HTT (0.33)
SCHEMBL20317403 0.79 CACNA1I (0.40) OPRL1
SCHEMBL25877203 0.79 ARG1 (0.41) ARG1ARG2CHRM4NOS3NOS1
SCHEMBL23105099 0.78 ARG1 (0.40) ARG1ARG2CHRM4NOS3NOS1
SCHEMBL25915237 0.78 HTT (0.32)
SCHEMBL25848264 0.76
SCHEMBL23594363 0.76 ATM (0.31)
SCHEMBL26805516 0.76 HRH3 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200339572-A1 NOVEL SELECTIVE CDK4/6 INHIBITOR AND PREPARATION THEREOF WUXI SHUANGLIANG BIOTECHNOLOGY CO., LTD. (CN) 2020-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200339572-A1 NOVEL SELECTIVE CDK4/6 INHIBITOR AND PREPARATION THEREOF CDK4, CDK6, CCNI ARG1 4008/4885ARG2 4629/4885CHRM4 2918/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.