SCHEMBL22604693

SCHEMBL22604693

O=C(N[C@H](Cc1ccc(Cl)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O)c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.62
PTPN1 P18031 3/20 0.62
CTSL P07711 4/20 0.60
ACE P12821 4/20 0.60
CTSS P25774 2/20 0.57
CTSK P43235 2/20 0.57
CA1 P00915 1/20 0.56
PSMB5 P28074 2/20 0.55
CTSV O60911 1/20 0.55
CTSB P07858 1/20 0.55
MME P08473 3/20 0.55
GPR132 Q9UNW8 1/20 0.54
CPA1 P15085 2/20 0.53
ACE2 Q9BYF1 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27679107 0.96 CTSL (0.64) CA2PTPN1CTSLACECTSS
SCHEMBL4359915 0.96 CTSL (0.64) CA2PTPN1CTSLACECTSS
SCHEMBL4369316 0.95 CTSL (0.63) CA2PTPN1CTSLACECTSS
SCHEMBL4357736 0.92 ACE (0.68) CA2PTPN1CTSLACECTSS
SCHEMBL4356229 0.92 ACE (0.68) CA2PTPN1CTSLACECTSS
SCHEMBL1305154 0.90 PTPN1 (0.70) CA2PTPN1CTSLACECA1
SCHEMBL8510030 0.90 PTPN1 (0.70) CA2PTPN1CTSLACECA1
SCHEMBL28760302 0.88 CTSL (0.67) CA2PTPN1CTSLACECTSS
SCHEMBL4369236 0.88 CTSL (0.67) CA2PTPN1CTSLACECTSS
SCHEMBL13669589 0.88 CTSL (0.67) CA2PTPN1CTSLACECTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020216240-A1 DICYCLIC ALKANE COMPOUND USEFUL AS INHIBITOR OF PLASMA KALLIKREIN 南京明德新药研发有限公司 2020-10-29 WO disclosed